SCHEMBL4978680

SCHEMBL4978680

Cc1nc(C(F)(F)C(F)(F)F)ccc1N

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.34
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
ALDH1A1 P00352 1/20 0.32
PRMT6 Q96LA8 1/20 0.31
KDM4E B2RXH2 1/20 0.30
CXCR4 P61073 1/20 0.30
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29626748 0.83 HSP90AA1 (0.44) HSP90AA1HSP90AB1ALDH1A1PRMT6KDM4E
SCHEMBL180808 0.83 HSP90AA1 (0.44) HSP90AA1HSP90AB1ALDH1A1PRMT6KDM4E
SCHEMBL6293989 0.76 NOS3 (0.34) HSP90AA1HSP90AB1NOS3NOS1NOS2
SCHEMBL2068476 0.73 SMN1; SMN2 (0.32) SMN1; SMN2NOS3NOS1NOS2
SCHEMBL1831943 0.68 SMN1; SMN2 (0.31) SMN1; SMN2
SCHEMBL3257531 0.68 ALDH1A1 (0.37) SMN1; SMN2HSP90AA1ALDH1A1KDM4E
SCHEMBL29686176 0.67
SCHEMBL2067821 0.67
SCHEMBL1653770 0.66
SCHEMBL31105996 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080045727-A1 Chiral 3-Halophthalic Acid Derivatives BAYER CROPSCIENCE AG (DE) 2008-02-21 US disclosed
EP-1789383-A1 CHIRAL 3-HALOPHTHALIC ACID DERIVATIVES Bayer CropScience AG (DE) 2007-05-30 EP disclosed
WO-2006024402-A1 CHIRAL 3-HALOPHTHALIC ACID DERIVATIVES BAYER CROPSCIENCE AG (DE) 2006-03-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080045727-A1 Chiral 3-Halophthalic Acid Derivatives HDHD5, CRYZ, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 SMN1; SMN2 4855/4885HSP90AA1 867/4885HSP90AB1 1289/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.