SCHEMBL4978701

SCHEMBL4978701

CC(C)(C)N(C(=O)O)C1CC1(Cc1ccncc1)S(N)(=O)=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.34
HTT P42858 2/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
RECQL P46063 2/20 0.33
PKM P14618 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KDM4E B2RXH2 1/20 0.32
CYP19A1 P11511 5/20 0.32
NAMPT P43490 4/20 0.32
CYP17A1 P05093 2/20 0.31
CA2 P00918 2/20 0.30
P2RX7 Q99572 1/20 0.30
CA1 P00915 1/20 0.30
CA5A P35218 1/20 0.30
CA7 P43166 1/20 0.30
CA5B Q9Y2D0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4978747 0.86 RIPK1 (0.34) MEN1KMT2A
SCHEMBL4977504 0.84 TAS2R14 (0.38) ALDH1A1KMT2ACA2CA1CA5A
SCHEMBL4977208 0.81 ALDH1A1 (0.37) ALDH1A1GAAKMT2AKDM4ECA2
SCHEMBL4981384 0.77 ALDH1A1 (0.36) ALDH1A1MEN1GAAKMT2APKM
SCHEMBL6050979 0.77 CYP19A1 (0.34) ALDH1A1HTTSMN1; SMN2RECQLPKM
SCHEMBL4983526 0.76 EPHX2 (0.35) ALDH1A1GAA
SCHEMBL4984750 0.74 MEN1 (0.36) ALDH1A1MEN1GAAKMT2ACA2
SCHEMBL4975355 0.74 MEN1 (0.36) ALDH1A1HTTMEN1GAAKMT2A
SCHEMBL4977363 0.74
SCHEMBL4978610 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1505945-B1 SUBSTITUTED CYCLOALKYL P1' HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2008-11-05 EP disclosed
US-6878722-B2 Substituted cycloalkyl P1′ hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2005-04-12 US disclosed
US-20040077551-A1 Substituted cycloalkyl P1' hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY 2004-04-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040077551-A1 Substituted cycloalkyl P1' hepatitis C virus inhibitors HAVCR2, ANPEP, ENPEP ALDH1A1 2672/4885HTT 3541/4885MEN1 4174/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.