SCHEMBL4980340

SCHEMBL4980340

O=c1[nH]c2cc(-c3ncccc3CN(c3cccnc3)c3cccnc3)ccc2n1CC(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 14/20 0.39
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
GRIN1 Q05586 3/20 0.35
GRIN2B Q13224 3/20 0.35
EPHX2 P34913 1/20 0.34
KCNA5 P22460 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4979261 0.85 NOS3 (0.39) NOS3NOS1NOS2
SCHEMBL1367775 0.70 AR (0.36) METAP2NOS3NOS1NOS2KCNA5
SCHEMBL4980354 0.69 NOS3 (0.36) NOS3NOS1NOS2KCNA5
SCHEMBL18464810 0.68 DAO (0.43) METAP2
SCHEMBL1370175 0.67 GABRP (0.42) NOS3NOS1NOS2KCNA5
SCHEMBL14992944 0.62 METAP2 (0.46) METAP2
SCHEMBL4175626 0.62 MEN1 (0.62)
SCHEMBL29695485 0.62 MEN1 (0.62)
SCHEMBL10146587 0.62 METAP2 (0.46) METAP2
SCHEMBL1367397 0.60 NOS3 (0.35) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993551-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-11-26 EP claimed
WO-2007089735-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO claimed