SCHEMBL4979261

SCHEMBL4979261

Cn1c(=O)[nH]c2cc(-c3ncccc3CN(c3cccnc3)c3cccnc3)ccc21

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
KMO O15229 1/20 0.39
LMNA P02545 1/20 0.38
MAPK14 Q16539 2/20 0.37
MAPT P10636 4/20 0.36
PDE10A Q9Y233 1/20 0.35
MAOB P27338 1/20 0.35
DYRK1A Q13627 1/20 0.35
TP53 P04637 2/20 0.34
JAK1 P23458 1/20 0.34
JAK3 P52333 1/20 0.34
PDK1 Q15118 1/20 0.34
DRD1 P21728 1/20 0.33
PGR P06401 1/20 0.33
SYK P43405 1/20 0.33
PRKDC P78527 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4980340 0.85 METAP2 (0.39) NOS3NOS1NOS2
SCHEMBL4980354 0.73 NOS3 (0.36) NOS3NOS1NOS2PDK1PRKDC
SCHEMBL1370175 0.71 GABRP (0.42) NOS3NOS1NOS2LMNAMAPT
SCHEMBL1367495 0.68 PRKDC (0.35) NOS3NOS1NOS2PDE10APRKDC
SCHEMBL1367397 0.66 NOS3 (0.35) NOS3NOS1NOS2PRKDC
SCHEMBL1369269 0.64 NOS2 (0.42) NOS3NOS1NOS2MAOBPRKDC
SCHEMBL1369018 0.63 CYP17A1 (0.46)
SCHEMBL1367302 0.63 KCNA5 (0.64) NOS3NOS1NOS2PRKDC
SCHEMBL4312246 0.63 DAO (0.50) LMNAMAPTPGR
SCHEMBL30176622 0.62 KMT2A (0.55) LMNAJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993551-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-11-26 EP disclosed
WO-2007089735-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO disclosed