SCHEMBL4980427

SCHEMBL4980427

NS(=O)(=O)C1(Cc2ncoc2-c2ccccc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LIMK2 P53671 1/20 0.42
ADORA2A P29274 1/20 0.41
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
FBP1 P09467 1/20 0.34
SCN9A Q15858 1/20 0.33
CA1 P00915 4/20 0.31
CA2 P00918 4/20 0.31
CA12 O43570 3/20 0.31
CA9 Q16790 3/20 0.31
KLKB1 P03952 1/20 0.31
PTGS2 P35354 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4977425 0.87 IMPDH2 (0.38) LIMK2ADORA2AHCRTR1HCRTR2FBP1
SCHEMBL4977420 0.74 LIMK2 (0.36) LIMK2ADORA2AHCRTR1HCRTR2FBP1
SCHEMBL4937409 0.74 LIMK2 (0.47) LIMK2ADORA2AHCRTR1HCRTR2FBP1
SCHEMBL4937416 0.71 LIMK2 (0.47) LIMK2ADORA2AHCRTR1HCRTR2FBP1
SCHEMBL635599 0.69 MAOA (0.50) CA1CA2CA12CA9MAOA
SCHEMBL4980952 0.69 TDO2 (0.53) CA1CA2CA12CA9PTGS2
SCHEMBL3075748 0.68 ADORA2A (0.50) LIMK2ADORA2AHCRTR1HCRTR2FBP1
SCHEMBL244662 0.68 ADORA2A (0.46) LIMK2ADORA2AHCRTR1HCRTR2FBP1
SCHEMBL2413968 0.68 ADORA2A (0.46) LIMK2ADORA2AHCRTR1HCRTR2FBP1
SCHEMBL14391718 0.68 ADORA2A (0.46) LIMK2ADORA2AHCRTR1HCRTR2FBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1505945-B1 SUBSTITUTED CYCLOALKYL P1' HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2008-11-05 EP disclosed
EP-1505945-A4 SUBSTITUTED CYCLOALKYL P1' HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2006-11-22 EP disclosed
US-6878722-B2 Substituted cycloalkyl P1′ hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2005-04-12 US disclosed
EP-1505945-A2 SUBSTITUTED CYCLOALKYL P1' HEPATITIS C VIRUS INHIBITORS Bristol-Myers Squibb Pharma Company (US) 2005-02-16 EP disclosed
WO-2004043339-A2 SUBSTITUTED CYCLOALKYL P1' HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-05-27 WO disclosed
WO-2004043339-A2 SUBSTITUTED CYCLOALKYL P1' HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-05-27 WO disclosed
US-20040077551-A1 Substituted cycloalkyl P1' hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY 2004-04-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040077551-A1 Substituted cycloalkyl P1' hepatitis C virus inhibitors HAVCR2, ANPEP, ENPEP LIMK2 4492/4885ADORA2A 3946/4885HCRTR1 2520/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.