Methapyrilene

Methapyrilene

SCHEMBL498484

CN(C)CCN(Cc1cccs1)c1ccccn1.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Methapyrilene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 3/20 0.97
KDM4E B2RXH2 4/20 1.00
KMT2A Q03164 4/20 1.00
MEN1 O00255 3/20 1.00
NPSR1 Q6W5P4 1/20 1.00
CYP2D6 P10635 6/20 0.97
CHRM2 P08172 4/20 0.97
ADRA2A P08913 4/20 0.97
DRD1 P21728 4/20 0.97
SLC6A4 P31645 4/20 0.97
SLC6A3 Q01959 4/20 0.97
KCNH2 Q12809 4/20 0.97
SLC6A2 P23975 3/20 0.97
HTR2A P28223 3/20 0.97
CYP1A2 P05177 3/20 0.97
OPRM1 P35372 3/20 0.97
ADRA2B P18089 2/20 0.97
CHRM1 P11229 2/20 0.97
HTR2C P28335 2/20 0.97
HTR2B P41595 2/20 0.97

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methapyrilene SCHEMBL19209 0.99 CYP2D6 (1.00) KDM4EKMT2AMEN1NPSR1CYP2D6
Methapyrilene SCHEMBL745149 0.97 CYP2D6 (0.97) KDM4EKMT2AMEN1NPSR1CYP2D6
Methapyrilene SCHEMBL1074644 0.96 CYP2D6 (0.95) KDM4EKMT2AMEN1NPSR1CYP2D6
Methapyrilene SCHEMBL7121305 0.91 CYP2D6 (0.86) KDM4EKMT2AMEN1NPSR1CYP2D6
Methapyrilene SCHEMBL28140755 0.91 CYP2D6 (0.86) KDM4EKMT2AMEN1NPSR1CYP2D6
Methapyrilene SCHEMBL4902232 0.88 CYP2D6 (0.80) KDM4EKMT2AMEN1NPSR1CYP2D6
SCHEMBL7297232 0.83 CYP2D6 (0.73) KDM4EKMT2AMEN1NPSR1CYP2D6
SCHEMBL10674626 0.81 CYP2D6 (0.70) KDM4EKMT2AMEN1NPSR1CYP2D6
SCHEMBL7311717 0.80 CYP2D6 (0.68) KDM4EKMT2AMEN1NPSR1CYP2D6
Histapyrrodine SCHEMBL28086254 0.79 HRH1 (0.64) KDM4EKMT2AMEN1NPSR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3593 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4742350-A1 ELECTROLYTE FOR LITHIUM SECONDARY BATTERY AND LITHIUM SECONDARY BATTERY INCLUDING THE SAME SK On Co., Ltd. (KR) 2026-05-13 EP claimed
US-20260112700-A1 Electrolyte for Lithium Secondary Battery and Lithium Secondary Battery Including the Same SK ON CO LTD (KR) 2026-04-23 US claimed
CN-113113521-B Light emitting device 三星显示有限公司 2025-03-28 CN claimed
CN-119294686-B Digital twinning-based shore power equipment management and control method and system 广州南沙海港集装箱码头有限公司 2025-03-25 CN claimed
CN-119462729-A Ladder alkenyl crosslinking comonomer, degradable PDCPD thermosetting material, preparation method and application 安徽建筑大学 2025-02-18 CN claimed
CN-119294686-A Digital twinning-based shore power equipment management and control method and system 广州南沙海港集装箱码头有限公司 2025-01-10 CN claimed
CN-117887009-A Preparation method and application of structure-controllable pigment hyper-dispersant 浙江纳美新材料股份有限公司 2024-04-16 CN claimed
CN-117792809-A Vehicle network management method, device, computer equipment and storage medium 中国第一汽车股份有限公司 2024-03-29 CN claimed
CN-117586781-A Liquid crystal composition, liquid crystal display element and application thereof 捷恩智株式会社 2024-02-23 CN claimed
CN-116970406-A Liquid crystal composition and liquid crystal element 捷恩智株式会社 2023-10-31 CN claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
WO-1998058685-A1 DERMAL ADHESIVE PLASTER SUITABLE FOR TREATING LOCALIZED CUTANEOUS AFFECTIONS LABORATORIO ITALIANO BIOCHIMICO FARMACEUTICO LISAPHARMA S.P.A. (IT) 1998-12-30 WO claimed
CN-1182798-A Method for producing natural abscisic acid by fungus fermentation CHENGDU INST BIOLOGY CAS (CN) 1998-05-27 CN claimed
CN-1118806-A Method for extracting oil from tea-oil seed by using additive ZHANG ZHIXIANG (CN) 1996-03-20 CN claimed
CN-1095107-A Seaweed beta-carotene production-agent increasing INST OCEANOLOGY CHINESE ACAD (CN) 1994-11-16 CN claimed
US-4654209-A NITROGLYCERINE PLUS STEROID, ANTIHISTAMINE, ANALGESIC, ANTIMICROBIAL EUROCELTIQUE, S.A. (LU) 1987-03-31 US claimed
US-4550067-A Secondary battery HITACHI, LTD. (JP) 1985-10-29 US claimed
US-4269835-A Nasal composition for relieving nasal distress WHITTLE BARRY J 1981-05-26 US claimed