Rigosertib

Rigosertib

SCHEMBL498623

COc1cc(OC)c(/C=C/S(=O)(=O)Cc2ccc(OC)c(NCC(=O)O)c2)c(OC)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 4/20 1.00
MET P08581 1/20 1.00
NQO2 P16083 1/20 1.00
FECH P22830 1/20 1.00
CLK3 P49761 1/20 1.00
HDAC3 O15379 2/20 0.81
HDAC4 P56524 2/20 0.81
HDAC1 Q13547 2/20 0.81
HDAC7 Q8WUI4 2/20 0.81
HDAC2 Q92769 2/20 0.81
HDAC10 Q969S8 2/20 0.81
HDAC11 Q96DB2 2/20 0.81
HDAC8 Q9BY41 2/20 0.81
HDAC6 Q9UBN7 2/20 0.81
HDAC9 Q9UKV0 2/20 0.81
HDAC5 Q9UQL6 2/20 0.81
MAPT P10636 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.40
ALDH1A1 P00352 3/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rigosertib SCHEMBL29397572 1.00 PLK1 (1.00) PLK1METNQO2FECHCLK3
Rigosertib SCHEMBL498624 1.00 PLK1 (1.00) PLK1METNQO2FECHCLK3
Rigosertib SCHEMBL498728 0.99 PLK1 (0.98) PLK1METNQO2FECHCLK3
Rigosertib SCHEMBL498730 0.99 PLK1 (0.98) PLK1METNQO2FECHCLK3
SCHEMBL25053516 0.93 PLK1 (0.87) PLK1METNQO2FECHCLK3
SCHEMBL4556188 0.93 PLK1 (0.87) PLK1METNQO2FECHCLK3
SCHEMBL6072521 0.93 PLK1 (0.87) PLK1METNQO2FECHCLK3
SCHEMBL498447 0.92 PLK1 (0.84) PLK1METNQO2FECHCLK3
SCHEMBL498448 0.92 PLK1 (0.84) PLK1METNQO2FECHCLK3
SCHEMBL12324480 0.92 PLK1 (0.84) PLK1METNQO2FECHCLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1721 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122057044-A Nanometer liposome delivery system for targeting PLK1/Aurora kinase and application thereof in oral squamous cell carcinoma treatment 徐州医科大学 2026-05-19 CN claimed
EP-4735445-A1 KRAS MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2026-05-06 EP claimed
EP-4735453-A1 KRAS MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2026-05-06 EP claimed
US-12616671-B2 Use of rigosertib to treat RNA virus infections ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2026-05-05 US claimed
EP-4363043-B1 COMPOSITIONS FOR USE IN METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2026-04-22 EP claimed
EP-4729519-A1 CRYSTAL FORM OF ENPP1 INHIBITOR CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang) Co., Ltd. (CN) 2026-04-22 EP claimed
US-12594421-B2 Compositions and methods for increasing cancer cell sensitivity to alternating electric fields NOVOCURE GMBH (CH) 2026-04-07 US claimed
US-20260092327-A1 METHODS OF MONITORING MUTATIONS IN TREATMENT OF COLORECTAL CANCER CARDIFF ONCOLOGY INC (US) 2026-04-02 US claimed
US-20260076970-A1 CANCER TREATMENT USING MTDP INHIBITORS AND PLK1 INHIBITORS CARDIFF ONCOLOGY INC (US) 2026-03-19 US claimed
US-20260053761-A1 USE OF THYROMIMETICS FOR THE TREATMENT OF CANCER UNIV OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2026-02-26 US claimed
US-20080161252-A1 Composition and Methods For the Treatment of Proliferative Diseases TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2008-07-03 US claimed
WO-2008027049-A1 COMPOSITION AND METHODS FOR THE TREATMENT OF MYELODYSPLASTIC SYNDROME AND ACUTE MYELOID LEUKEMIA TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2008-03-06 WO claimed
EP-1773353-A2 FORMULATIONS FOR PARENTERAL ADMINISTRATION OF (E)-2,6-DIALKOXYSTRYRYL 4-SUBSTITUTED BENZYLSULFONES Onconova Therapeutics, Inc (US) 2007-04-18 EP claimed
WO-2006104668-A2 COMPOSITION AND METHODS FOR THE TREATMENT OF PROLIFERATIVE DISEASES TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2006-10-05 WO claimed
EP-1487428-A4 AMINO-SUBSTITUTED (E)-2,6-DIALKOXYSTYRYL 4-SUBSTITUTED BENZYLSULFONES FOR TREATING PROLIFERATIVE DISORDERS UNIV TEMPLE (US) 2006-04-19 EP claimed
WO-2006010152-A2 FORMULATIONS FOR PARENTERAL ADMINISTRATION OF (E)-2,6-DIALKOXYSTRYRYL 4-SUBSTITUTED BENZYLSULFONES ONCONOVA THERAPEUTICS, INC. (US) 2006-01-26 WO claimed
WO-2005065074-A2 PROTECTION OF TISSUES AND CELLS FROM CYTOTOXIC EFFECTS OF IONIZING RADIATION BY ABL INHIBITORS TEMPLE UNIVERSITY OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2005-07-21 WO claimed
US-20050130942-A1 Amino-substituted (e)-2,6-dialkoxystyryl 4-substituted-benzylsulfones for treating proliferative disorders TEMPLE UNIVERSITY OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2005-06-16 US claimed
EP-1487428-A2 AMINO-SUBSTITUTED (E)-2,6-DIALKOXYSTYRYL 4-SUBSTITUTED BENZYLSULFONES FOR TREATING PROLIFERATIVE DISORDERS Temple University of the Commonwealth System of Higher Education (US) 2004-12-22 EP claimed
WO-2003072062-A2 AMINO-SUBSTITUTED (E)-2,6-DIALKOXYSTYRYL 4-SUBSTITUTED BENZYLSULFONES FOR TREATING PROLIFERATIVE DISORDERS TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2003-09-04 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161252-A1 Composition and Methods For the Treatment of Proliferative Diseases CCNH, POLH, CCNO PLK1 196/4885MET 254/4885NQO2 733/4885
US-20260076970-A1 CANCER TREATMENT USING MTDP INHIBITORS AND PLK1 INHIBITORS PLK1, PLK4, PLK2 PLK1 1/4885MET 269/4885NQO2 3366/4885
US-12616671-B2 Use of rigosertib to treat RNA virus infections EIF2AK2, ACE2, SARS1 PLK1 91/4885MET 1545/4885NQO2 1273/4885
US-12594421-B2 Compositions and methods for increasing cancer cell sensitivity to alternating electric fields PTK2, GSK3B, MTOR PLK1 68/4885MET 724/4885NQO2 3408/4885
US-20260053761-A1 USE OF THYROMIMETICS FOR THE TREATMENT OF CANCER THRA, THRB, TRHR PLK1 2636/4885MET 292/4885NQO2 1524/4885
US-20260092327-A1 METHODS OF MONITORING MUTATIONS IN TREATMENT OF COLORECTAL CANCER KRAS, HRAS, NRAS PLK1 25/4885MET 136/4885NQO2 2185/4885
US-20050130942-A1 Amino-substituted (e)-2,6-dialkoxystyryl 4-substituted-benzylsulfones for treating proliferative disorders CCNY, CCND2, CCNB1 PLK1 1376/4885MET 1078/4885NQO2 151/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.