SCHEMBL5009841

SCHEMBL5009841

CC(C)(O)c1ccc(-c2ccc(CC=O)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.38
RXRB P28702 2/20 0.38
RXRG P48443 2/20 0.38
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
TNKS O95271 9/20 0.35
PARP1 P09874 9/20 0.35
TNKS2 Q9H2K2 9/20 0.35
CDC7 O00311 1/20 0.35
PLK4 O00444 1/20 0.35
CHEK1 O14757 1/20 0.35
AURKA O14965 1/20 0.35
PDPK1 O15530 1/20 0.35
JAK2 O60674 1/20 0.35
MAP4K4 O95819 1/20 0.35
PAK4 O96013 1/20 0.35
CHEK2 O96017 1/20 0.35
ABL1 P00519 1/20 0.35
LCK P06239 1/20 0.35
FYN P06241 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1427894 0.94 TP53 (0.40) TP53TSHRCCR9ESR1ESR2
SCHEMBL5011507 0.83 BCL2 (0.45) RXRARXRB
SCHEMBL13974830 0.79 EGFR (0.44) RXRARXRBRXRGTP53CDC7
SCHEMBL18802754 0.78 KIF11 (0.44) TSHRTNKSPARP1TNKS2CDC7
SCHEMBL547767 0.78 KIF11 (0.44) TSHRTNKSPARP1TNKS2CDC7
SCHEMBL3392101 0.78 HRH3 (0.43) RXRARXRBRXRGTSHR
SCHEMBL3639494 0.77 TSHR (0.57) TP53TSHREPHX2NR1H4
Hydrochloric Acid SCHEMBL21352581 0.76 HRH3 (0.41) TSHR
SCHEMBL1428666 0.76 ALDH1A1 (0.48) TP53TSHRTNKSPARP1ESR1
SCHEMBL2267819 0.76 KIF11 (0.55) RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP claimed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO claimed