SCHEMBL5012369

SCHEMBL5012369

C=C(CC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.39
MAOB P27338 6/20 0.39
CES1 P23141 1/20 0.34
ESR1 P03372 1/20 0.33
CA2 P00918 1/20 0.33
POLB P06746 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14123664 1.00 MAOA (0.39) MAOAMAOBCES1ESR1CA2
SCHEMBL5008736 1.00 MAOA (0.39) MAOAMAOBCES1ESR1CA2
SCHEMBL7792771 0.98 MAOA (0.40) MAOAMAOBCES1ESR1CA2
SCHEMBL7791505 0.93 MAOA (0.41) MAOAMAOBCES1ESR1POLB
SCHEMBL7790765 0.79 MAOA (0.37) MAOAMAOBCES1ESR1POLB
SCHEMBL7792764 0.77 ESR1 (0.47) MAOAMAOBCES1ESR1CYP3A4
SCHEMBL8396822 0.76 MAOA (0.42) MAOAMAOBCES1ESR1POLB
SCHEMBL7783038 0.75 MAOA (0.39) MAOAMAOBCES1ESR1NPSR1
SCHEMBL8624256 0.74 MAOA (0.33) MAOAMAOB
SCHEMBL20690145 0.74 MAOA (0.42) MAOAMAOBCES1CA2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080194887-A1 SEPARATION OF FLUOROUS COMPOUNDS PITTSBURGH UNIVERSITY OF - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2008-08-14 US disclosed
US-7364908-B2 Separation of fluorous compounds UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2008-04-29 US disclosed
EP-1765783-A1 SEPARATION OF FLUOROUS COMPOUNDS UNIVERSITY OF PITTSBURGH (US) 2007-03-28 EP disclosed
WO-2006009835-A1 SEPARATION OF FLUOROUS COMPOUNDS UNIVERSITY OF PITTSBURGH (US) 2006-01-26 WO disclosed
US-20050283032-A1 charging a mixture of compounds to a non-fluorous solid phase (silica gel, alumina, zirconia) and eluting with a fluorous eluting fluid (hydrofluoroalkane, a hydrofluoroether, a hydrofluoroamine, a perfluoroalkane, a perfluoroether, or a perfluoroamine) and a cosolvent: difference in fluorous nature NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2005-12-22 US disclosed