SCHEMBL5012881

SCHEMBL5012881

C=CCNC(=S)N1N(Cc2ccc3ccccc3c2)C(=O)OC12CCCCC2

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
IDO1 P14902 1/20 0.34
FAAH O00519 4/20 0.34
POLB P06746 1/20 0.33
MAPT P10636 3/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MMP13 P45452 1/20 0.33
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33
MAPK1 P28482 1/20 0.33
ACHE P22303 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GRM1 Q13255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1086672 0.75 KDM4E (0.44) KDM4EALDH1A1L3MBTL1FAAHPOLB
SCHEMBL9400347 0.63 NR1H4 (0.56) ALDH1A1L3MBTL1MAPTGAAHPGD
SCHEMBL5012778 0.60 TP53 (0.37) ALDH1A1LMNAKMT2A
SCHEMBL4486194 0.59 TACR2 (0.41) FAAHMMP13PKMKMT2A
SCHEMBL7357694 0.58 GRM1 (0.46) ACHEGRM1
SCHEMBL11558110 0.57 NR1H4 (0.39) L3MBTL1IDO1GAAMEN1KMT2A
SCHEMBL7357166 0.56 GRM1 (0.45) ACHEGRM1
SCHEMBL31010303 0.56 KMT2A (0.74) ALDH1A1POLBPKMACHEKMT2A
SCHEMBL5195380 0.56 KMT2A (0.74) ALDH1A1POLBPKMACHEKMT2A
SCHEMBL3383094 0.56 L3MBTL1 (0.69) L3MBTL1MMP13PKMACHEKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed