SCHEMBL5012930

SCHEMBL5012930

N#Cc1ccc(CN2C(=O)OC3(CCCCC3)N2C(=O)c2cccc(Cl)c2Cl)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.38
CNR1 P21554 1/20 0.38
MDM2 Q00987 3/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
PGGT1B P53609 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
CYP2C19 P33261 5/20 0.36
MAPK1 P28482 3/20 0.36
CYP3A4 P08684 8/20 0.36
USP2 O75604 6/20 0.36
ALDH1A1 P00352 5/20 0.36
CYP1A2 P05177 4/20 0.36
CYP2C9 P11712 4/20 0.36
P2RX7 Q99572 1/20 0.36
CYP2D6 P10635 4/20 0.35
TSHR P16473 3/20 0.35
TP53 P04637 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5013344 0.82 CNR2 (0.38) CNR2CNR1CYP2C19MAPK1CYP3A4
SCHEMBL5016264 0.79 HPGD (0.38) CNR2CNR1CYP2C19MAPK1CYP3A4
SCHEMBL5170031 0.75 MAPK14 (0.49) MAPK1ALDH1A1
SCHEMBL1086471 0.74 CYP2C19 (0.45) TRPM8CYP2C19MAPK1CYP3A4USP2
SCHEMBL5013547 0.70 POLB (0.39) CNR2CYP2C19CYP3A4ALDH1A1CYP1A2
SCHEMBL5012929 0.66 HPGD (0.40) CNR2CNR1HPGD
SCHEMBL1086521 0.61 CYP3A4 (0.48) TRPM8CYP2C19MAPK1CYP3A4USP2
SCHEMBL3077014 0.61 GRM2 (0.52) CYP2C19CYP3A4USP2ALDH1A1CYP1A2
SCHEMBL29944015 0.59 HPGD (0.67) USP2P2RX7GLAMEN1KMT2A
SCHEMBL26037565 0.58 ALDH1A1 (0.68) MAPK1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed