SCHEMBL5013344

SCHEMBL5013344

N#Cc1ccc(CN2C(=O)OC3(CCCCC3)N2C(=O)c2ccc(Cl)c(Cl)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.38
CNR1 P21554 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 10/20 0.38
USP2 O75604 6/20 0.38
CYP2D6 P10635 5/20 0.38
ALDH1A1 P00352 4/20 0.37
CYP1A2 P05177 3/20 0.37
CYP2C19 P33261 3/20 0.37
ABCC9 O60706 1/20 0.37
GLA P06280 1/20 0.37
CYP2C9 P11712 4/20 0.37
TSHR P16473 3/20 0.37
HPGD P15428 2/20 0.37
MAPK1 P28482 2/20 0.37
FASN P49327 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5012930 0.82 CNR2 (0.38) CNR2CNR1CYP3A4USP2CYP2D6
SCHEMBL5016264 0.76 HPGD (0.38) CNR2CNR1CYP3A4USP2CYP2D6
SCHEMBL1087047 0.73 CYP3A4 (0.48) POLBCYP3A4USP2CYP2D6ALDH1A1
SCHEMBL5170031 0.71 MAPK14 (0.49) POLBALDH1A1MAPK1LMNA
SCHEMBL5011733 0.68 EPHX2 (0.39) CYP3A4ALDH1A1CYP2C9TSHRHPGD
SCHEMBL5013591 0.67 TSHR (0.47) POLBCYP3A4USP2CYP2D6ALDH1A1
SCHEMBL5012907 0.65 TSHR (0.46) ALDH1A1TSHRHPGDSMN1; SMN2LMNA
SCHEMBL5012929 0.63 HPGD (0.40) CNR2CNR1HPGDLMNAHTT
SCHEMBL3568071 0.62 MAPT (0.47) ALDH1A1HPGDLMNAHTT
SCHEMBL3077014 0.61 GRM2 (0.52) CYP3A4USP2CYP2D6ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed