SCHEMBL5013547

SCHEMBL5013547

Cc1cc(C(=O)N2N(Cc3cccc(C#N)c3)C(=O)OC23CCCCC3)no1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CNR2 P34972 2/20 0.37
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
ACKR3 P25106 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PARG Q86W56 2/20 0.36
TAS2R8 Q9NYW2 2/20 0.36
FAAH O00519 1/20 0.36
CYP1A2 P05177 3/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
KLKB1 P03952 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011708 0.87 CYP1A2 (0.45) NPC1RAB9AACKR3KDM4EALDH1A1
SCHEMBL5012778 0.81 TP53 (0.37) NPC1RAB9AALDH1A1
SCHEMBL5066991 0.76 RAB9A (0.38) NPC1RAB9AKDM4EALDH1A1CYP1A2
SCHEMBL1087064 0.76 KMT2A (0.43) POLBRXFP1NPC1RAB9ASIRT2
SCHEMBL5012930 0.70 CNR2 (0.38) CNR2ALDH1A1CYP1A2CYP3A4TSHR
SCHEMBL5013344 0.69 CNR2 (0.38) POLBCNR2ALDH1A1CYP1A2CYP3A4
SCHEMBL5011651 0.67 CHRM2 (0.44) KDM4EALDH1A1TSHR
SCHEMBL5011764 0.65 HTT (0.44) CNR2ALDH1A1TSHR
SCHEMBL1086550 0.60 TSHR (0.49) NPC1RAB9AALDH1A1CYP1A2CYP3A4
SCHEMBL7359317 0.60 KLKB1 (0.51) POLBKDM4EALDH1A1PARGKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed