SCHEMBL5012907

SCHEMBL5012907

Cc1ccc(CN2C(=O)OC3(CCCCC3)N2OC(=O)NCc2ccc(Cl)c(Cl)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ERN1 O75460 1/20 0.43
LMNA P02545 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HPGD P15428 1/20 0.40
ESR1 P03372 1/20 0.39
NR3C1 P04150 1/20 0.39
PGR P06401 1/20 0.39
NR3C2 P08235 1/20 0.39
ESR2 Q92731 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
TAOK1 Q7L7X3 2/20 0.37
TAOK3 Q9H2K8 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
THRB P10828 1/20 0.37
P2RX7 Q99572 1/20 0.37
CHRM2 P08172 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011798 0.88 TSHR (0.41) TSHRSMN1; SMN2LMNAALDH1A1HTT
SCHEMBL5011597 0.80 PLAAT3 (0.41) SMN1; SMN2LMNAALDH1A1EPHX2
SCHEMBL4272713 0.75 TSHR (0.45) TSHRSMN1; SMN2ERN1ALDH1A1HPGD
SCHEMBL5013516 0.74 RAB9A (0.46) SMN1; SMN2LMNAALDH1A1NPSR1HPGD
SCHEMBL1086318 0.67 ERN1 (0.54) TSHRSMN1; SMN2ERN1LMNAALDH1A1
SCHEMBL5012256 0.65 TP53 (0.46) TSHRLMNAALDH1A1THRBCHRM1
SCHEMBL9659041 0.65 TSHR (1.00) TSHRSMN1; SMN2LMNAALDH1A1HPGD
SCHEMBL5013344 0.65 CNR2 (0.38) TSHRSMN1; SMN2LMNAALDH1A1HTT
SCHEMBL5351946 0.64 CHRM2 (0.50) SMN1; SMN2ERN1ALDH1A1HTTNPSR1
SCHEMBL7616443 0.64 LMNA (0.65) TSHRSMN1; SMN2LMNAALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed