SCHEMBL5013432

SCHEMBL5013432

Cc1ccc(NC(=O)ON2N(Cc3ccc(SC(F)(F)F)cc3)C(=O)OC23CCCCC3)cc1[N+](=O)[O-]

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.40
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
KMT2A Q03164 8/20 0.37
ALDH1A1 P00352 5/20 0.37
HPGD P15428 2/20 0.37
MEN1 O00255 6/20 0.36
HTT P42858 1/20 0.36
NPC1 O15118 4/20 0.35
ALOX12 P18054 1/20 0.35
MAPT P10636 6/20 0.34
LMNA P02545 4/20 0.34
MAPK1 P28482 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
ATM Q13315 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
PPIA P62937 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5013516 0.89 RAB9A (0.46) RAB9AKMT2AALDH1A1HPGDMEN1
SCHEMBL5012911 0.80 PPARG (0.36) PPARGPPARAKMT2AALDH1A1HPGD
SCHEMBL4258712 0.80 PPARG (0.38) RAB9APPARGPPARAKMT2AALDH1A1
SCHEMBL5011711 0.72 MAPT (0.46) KMT2AALDH1A1MEN1HTTMAPT
SCHEMBL4262167 0.68 MAPT (0.43) RAB9AKMT2AALDH1A1HPGDMEN1
SCHEMBL4269518 0.66 ALDH1A1 (0.41) RAB9AKMT2AALDH1A1HPGDMEN1
SCHEMBL5011733 0.66 EPHX2 (0.39) KMT2AALDH1A1HPGDMEN1SMN1; SMN2
SCHEMBL1449040 0.63 MAPT (0.58) RAB9AKMT2AALDH1A1HPGDMEN1
SCHEMBL10889357 0.62 KMT2A (0.65) RAB9AKMT2AALDH1A1HPGDMEN1
SCHEMBL12708550 0.62 ALDH1A1 (0.50) RAB9AKMT2AALDH1A1MEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed