SCHEMBL5011764

SCHEMBL5011764

Cc1ccc(C(=O)N2N(Cc3ccccc3)C(=O)OC23CCCCC3)c(F)c1F

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.44
HPGD P15428 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
THRB P10828 1/20 0.34
AGTR1 P30556 3/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
CACNA1G O43497 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5012929 0.90 HPGD (0.40) HTTHPGDL3MBTL1CNR1CNR2
SCHEMBL5016264 0.88 HPGD (0.38) HPGDCNR1CNR2KMT2AMEN1
SCHEMBL5011708 0.76 CYP1A2 (0.45) HTTHPGDL3MBTL1KMT2ALMNA
SCHEMBL5013449 0.75 KAT6A (0.39)
SCHEMBL5011651 0.74 CHRM2 (0.44) L3MBTL1KMT2AMEN1LMNAALDH1A1
SCHEMBL1086210 0.72 HPGD (0.48) HTTHPGDL3MBTL1ALDH1A1TSHR
SCHEMBL5015150 0.71 MAPT (0.53) HTTKMT2AMEN1LMNAALDH1A1
SCHEMBL5011747 0.67 KCNK3 (0.40) HPGDKMT2ALMNAALDH1A1
SCHEMBL5016419 0.67 ALDH1A1 (0.41) HTTL3MBTL1LMNAALDH1A1TSHR
SCHEMBL5011879 0.67 KMT2A (0.38) HPGDKMT2AMEN1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed