SCHEMBL5015224

SCHEMBL5015224

FC(F)(F)c1ccccc1C=C1CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 2/20 0.51
IL6 P05231 2/20 0.51
HTR2C P28335 3/20 0.47
MYC P01106 1/20 0.46
MAX P61244 1/20 0.46
NFKB1 P19838 1/20 0.41
CCR3 P51677 1/20 0.39
CYP24A1 Q07973 1/20 0.39
GRIN2D O15399 2/20 0.38
GRIN3B O60391 2/20 0.38
GRIN1 Q05586 2/20 0.38
GRIN2A Q12879 2/20 0.38
GRIN2B Q13224 2/20 0.38
GRIN2C Q14957 2/20 0.38
GRIN3A Q8TCU5 2/20 0.38
EPHX2 P34913 1/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
MAOB P27338 1/20 0.36
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25375799 0.87 TNF (0.59) TNFIL6MYCMAXNFKB1
SCHEMBL12751291 0.77 IKBKB (0.51) HTR2CMAOB
Hydrochloric Acid SCHEMBL6979971 0.75 IKBKB (0.50) HTR2CGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8315728 0.74 PRCP (0.42) HTR2CSLC6A2SLC6A4
SCHEMBL12751382 0.73 HTR2C (0.47) HTR2CNFKB1MAOB
SCHEMBL12751389 0.73 DYRK2 (0.51) HTR2CMAOB
SCHEMBL12751376 0.73 HTR2C (0.45) HTR2CNFKB1
SCHEMBL28292786 0.73 LMNA (0.50) HTR2CMAOB
SCHEMBL28211553 0.72 MYC (0.49) TNFIL6HTR2CMYCMAX
SCHEMBL28211015 0.72 TNF (0.51) TNFIL6HTR2CMYCMAX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951731-A1 AZACYCLOHEXANE DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE Merck Frosst Canada Ltd. (CA) 2008-08-06 EP disclosed
WO-2007056846-A1 AZACYCLOHEXANE DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2007-05-24 WO disclosed