SCHEMBL28211015

SCHEMBL28211015

FC(F)(F)c1ccccc1C=C1CCCCN1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 3/20 0.51
IL6 P05231 3/20 0.51
MYC P01106 1/20 0.43
MAX P61244 1/20 0.43
NFKB1 P19838 1/20 0.38
CCR3 P51677 1/20 0.37
CYP24A1 Q07973 1/20 0.36
GRIN2D O15399 2/20 0.36
GRIN3B O60391 2/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
GRIN2B Q13224 2/20 0.36
GRIN2C Q14957 2/20 0.36
GRIN3A Q8TCU5 2/20 0.36
LMNA P02545 1/20 0.35
HTR2C P28335 2/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8911935 0.82 RXRA (0.35) TNFIL6HPGDNPSR1MEN1
SCHEMBL28210997 0.78 TNF (0.51) TNFIL6MYCMAXNFKB1
SCHEMBL28211054 0.76 TNF (0.68) TNFIL6MYCMAXNFKB1
SCHEMBL1891515 0.76 TP53 (0.41) NFKB1LMNAHPGDMEN1CYP1A2
SCHEMBL1891513 0.76 TP53 (0.41) NFKB1LMNAHPGDMEN1CYP1A2
SCHEMBL5766522 0.76 HSD11B1 (0.47) CCR3MEN1KMT2A
SCHEMBL3855365 0.73 CYP26A1 (0.37) CCR3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL5015224 0.72 TNF (0.51) TNFIL6MYCMAXNFKB1
SCHEMBL28211553 0.72 MYC (0.49) TNFIL6MYCMAXNFKB1
SCHEMBL25375799 0.72 TNF (0.59) TNFIL6MYCMAXNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105037252-B N- substitutions -3,5- two (2- (trifluoromethyl) benzal) piperidin-4-one-derivative and preparation method and application 温州医科大学 2018-05-04 CN disclosed
CN-105037252-B N- substitutions -3,5- two (2- (trifluoromethyl) benzal) piperidin-4-one-derivative and preparation method and application 温州医科大学 2018-05-04 CN disclosed