SCHEMBL5016083

SCHEMBL5016083

COc1ccc(CN2CCN(c3cc([O])c4ncsc4c3)CC2)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
KDM4E B2RXH2 6/20 0.51
KMT2A Q03164 5/20 0.51
NPSR1 Q6W5P4 2/20 0.49
MAPT P10636 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
DRD2 P14416 3/20 0.48
DRD4 P21917 2/20 0.48
DRD3 P35462 2/20 0.48
TSHR P16473 2/20 0.47
ALOX15 P16050 1/20 0.47
MAPK1 P28482 3/20 0.45
LMNA P02545 2/20 0.45
HTT P42858 1/20 0.45
MEN1 O00255 3/20 0.44
TP53 P04637 1/20 0.44
PI4KB Q9UBF8 1/20 0.43
HSD17B10 Q99714 2/20 0.43
USP2 O75604 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5016084 0.89 ALDH1A1 (0.50) ALDH1A1KDM4EKMT2ANPSR1MAPT
SCHEMBL5011858 0.84 DRD4 (0.44) ALDH1A1KDM4EMAPTSMN1; SMN2DRD2
SCHEMBL2095343 0.84 ABCB1 (0.41) ALDH1A1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL27644661 0.83 DRD2 (0.52) ALDH1A1KDM4EKMT2ANPSR1MAPT
SCHEMBL5015139 0.78 PPARD (0.43) ALDH1A1KDM4ESMN1; SMN2DRD2DRD4
SCHEMBL5544192 0.76 ALDH1A1 (0.63) ALDH1A1KDM4EKMT2ANPSR1MAPT
SCHEMBL1600111 0.74 KMT2A (0.65) ALDH1A1KDM4EKMT2ATSHRALOX15
SCHEMBL5016097 0.73 KDM4E (0.44) ALDH1A1KDM4EMAPTDRD2DRD4
SCHEMBL5011868 0.72 DRD4 (0.41) ALDH1A1KDM4ENPSR1MAPTSMN1; SMN2
SCHEMBL5544199 0.71 ALDH1A1 (0.63) ALDH1A1KDM4EKMT2ANPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-B1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMA CO LTD (JP) 2008-10-08 EP disclosed