SCHEMBL5016897

SCHEMBL5016897

CC1CCC(NC(=O)O[C@@H]2C[C@@H]2CN2CCC(c3cc4ccccc4s3)CC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 7/20 0.47
DRD2 P14416 1/20 0.47
ALOX5 P09917 1/20 0.39
CNR1 P21554 6/20 0.37
CNR2 P34972 6/20 0.37
HTR1A P08908 4/20 0.37
HRH3 Q9Y5N1 1/20 0.36
SLC6A3 Q01959 2/20 0.36
RAB9A P51151 3/20 0.36
NPC1 O15118 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
CXCR6 O00574 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13201263 0.84 SLC6A4 (0.49) SLC6A4DRD2ALOX5CNR1CNR2
SCHEMBL5025700 0.72 TLR7 (0.36) DRD2
SCHEMBL5023889 0.70 HTR2A (0.40)
SCHEMBL5023353 0.70 HTR2A (0.48)
SCHEMBL11877556 0.68 SLC6A4 (0.70) SLC6A4DRD2ALOX5HTR1AHRH3
SCHEMBL5023775 0.67 DRD2 (0.37) DRD2HTR1ARAB9ANPC1
SCHEMBL5023822 0.67 DRD2 (0.36) DRD2HTR1ARAB9ANPC1
SCHEMBL6093432 0.66 RAB9A (0.60) DRD2HTR1ARAB9ANPC1SMN1; SMN2
SCHEMBL6093435 0.66 RAB9A (0.60) DRD2HTR1ARAB9ANPC1SMN1; SMN2
SCHEMBL11877235 0.66 DRD2 (0.60) SLC6A4DRD2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1632483-B1 HETEROCYCLIC SUBSTITUTED CARBONYL DERIVATIVES AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS AVENTIS PHARMA INC (US) 2008-10-29 EP claimed