SCHEMBL5023822

SCHEMBL5023822

CC1CCC(NC(=O)O[C@@H]2C[C@@H]2CN2CCN(c3nc4cccc5c4n3CCC5)CC2)CC1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.36
CYP11B2 P19099 1/20 0.32
DRD3 P35462 1/20 0.32
RAB9A P51151 4/20 0.32
NPC1 O15118 3/20 0.32
TSHR P16473 1/20 0.32
HTR1A P08908 2/20 0.31
HTR2A P28223 2/20 0.31
OPRD1 P41143 1/20 0.31
OPRL1 P41146 1/20 0.31
MCL1 Q07820 1/20 0.31
MAPT P10636 1/20 0.31
MEN1 O00255 1/20 0.30
USP2 O75604 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13201266 0.87 ALDH1A1 (0.35) DRD2DRD3RAB9ANPC1MAPT
SCHEMBL5023775 0.69 DRD2 (0.37) DRD2DRD3RAB9ANPC1HTR1A
SCHEMBL8544362 0.68 ALDH1A1 (0.47) NPC1TSHRMAPTMEN1USP2
SCHEMBL8543289 0.68 NPC1 (0.45) RAB9ANPC1MAPT
SCHEMBL8549930 0.67 MCL1 (0.46) RAB9ANPC1MCL1MAPTMEN1
SCHEMBL5016897 0.67 SLC6A4 (0.47) DRD2RAB9ANPC1HTR1A
SCHEMBL8545991 0.66 LMNA (0.50) DRD2DRD3RAB9ANPC1HTR1A
SCHEMBL8548519 0.65 MAPT (0.47) RAB9ANPC1TSHRMCL1MAPT
SCHEMBL8543387 0.64 HRH1 (0.45) DRD2DRD3RAB9ANPC1HTR1A
Hydrochloric Acid SCHEMBL8550810 0.64 MAPT (0.46) RAB9ANPC1TSHRMCL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1632483-B1 HETEROCYCLIC SUBSTITUTED CARBONYL DERIVATIVES AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS AVENTIS PHARMA INC (US) 2008-10-29 EP claimed