SCHEMBL5017358

SCHEMBL5017358

CCOC1(Br)C=CC(N)=CC1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2219369 0.79
SCHEMBL11687259 0.76
SCHEMBL5017147 0.75
SCHEMBL5023745 0.75
SCHEMBL334646 0.74
SCHEMBL13679854 0.69
SCHEMBL1331497 0.67 LTA4H (0.30)
SCHEMBL18856410 0.66
SCHEMBL20876924 0.66
SCHEMBL3670863 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250281433-A1 NOVEL DERIVATIVE COMPOUND HAVING BIPHENYL GROUP INTRODUCED INTO AMINO-ALKANOIC ACID AND ANTI-INFLAMMATORY COMPOSITION COMPRISING SAME AMTIXBIO CO., LTD. (KR) 2025-09-11 US disclosed
US-12180139-B2 Method for preparing aminoalkanoic acid derivative containing biphenyl group AMTIXBIO CO., LTD. (KR) 2024-12-31 US disclosed
US-12172945-B2 Aminoalkanoic acid derivative containing biphenyl group and use of the same AMTIXBIO CO., LTD. (KR) 2024-12-24 US disclosed
US-12129220-B2 Pharmaceutical composition comprising aminoalkanoic acid derivative containing biphenyl group AMTIXBIO CO., LTD. (KR) 2024-10-29 US disclosed
EP-3992177-B1 DERIVATIVE COMPOUND INTRODUCING BIPHENYL GROUP INTO NOVEL AMINOALKANOIC ACID AND ANTIFUNGAL PHARMACEUTICAL COMPOSITION COMPRISING SAME AMTIXBIO CO LTD (KR) 2024-05-08 EP disclosed
EP-4268811-A1 NOVEL DERIVATIVE COMPOUND HAVING BIPHENYL GROUP INTRODUCED INTO AMINO-ALKANOIC ACID AND ANTI-INFLAMMATORY COMPOSITION COMPRISING SAME Amtixbio Co., Ltd. (KR) 2023-11-01 EP disclosed
US-20230067422-A1 AMINOALKANOIC ACID DERIVATIVE CONTAINING BIPHENYL GROUP AND USE OF THE SAME AMTIXBIO CO., LTD. (KR) 2023-03-02 US disclosed
US-20230053855-A1 PHARMACEUTICAL COMPOSITION COMPRISING AMINOALKANOIC ACID DERIVATIVE CONTAINING BIPHENYL GROUP AMTIXBIO CO., LTD. (KR) 2023-02-23 US disclosed
US-20230056812-A1 METHOD FOR PREPARING AMINOALKANOIC ACID DERIVATIVE CONTAINING BIPHENYL GROUP AMTIXBIO CO., LTD. (KR) 2023-02-23 US disclosed
US-11479526-B2 Aminoalkanoic acid derivative containing biphenyl group and antifungal pharmaceutical composition comprising the same AMTIXBIO CO., LTD. (KR) 2022-10-25 US disclosed
US-20220144755-A1 NOVEL AMINOALKANOIC ACID DERIVATIVE CONTAINING BIPHENYL GROUP AND ANTIFUNGAL PHARMACEUTICAL COMPOSITION COMPRISING THE SAME AMTIXBIO CO., LTD. (KR) 2022-05-12 US disclosed
EP-3992177-A1 DERIVATIVE COMPOUND INTRODUCING BIPHENYL GROUP INTO NOVEL AMINOALKANOIC ACID AND ANTIFUNGAL PHARMACEUTICAL COMPOSITION COMPRISING SAME Amtixbio Co., Ltd. (KR) 2022-05-04 EP disclosed
US-20080268374-A1 Photosensitive Composition, Pattern Forming Material, Photosensitive Laminate, Pattern Forming Apparatus, and Pattern Forming Process FUJIFILM CORPORATION (JP) 2008-10-30 US disclosed
EP-1780599-A1 PHOTOSENSITIVE COMPOSITION, PATTERN FORMING MATERIAL, PHOTOSENSITIVE LAMINATE, PATTERN FORMING APPARATUS AND METHOD OF PATTERN FORMATION FUJIFILM Corporation (JP) 2007-05-02 EP disclosed