SCHEMBL5019111

SCHEMBL5019111

CN[C@@H](CC(=O)O)C(=O)OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
CASP1 P29466 12/20 0.51
HTT P42858 1/20 0.48
TACR1 P25103 1/20 0.47
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19511367 0.89 ALDH1A1 (0.53) ALDH1A1CASP1TACR1MAPK1L3MBTL1
SCHEMBL7753516 0.89 ALDH1A1 (0.53) ALDH1A1CASP1TACR1MAPK1L3MBTL1
SCHEMBL31276678 0.88 ABCB1 (0.51) ALDH1A1CASP1TACR1LMNAMAPK1
SCHEMBL29443514 0.86 CASP1 (0.48) ALDH1A1CASP1HTTLMNASMN1; SMN2
SCHEMBL8351818 0.85 ALDH1A1 (0.53) ALDH1A1TACR1LMNASMN1; SMN2MAPK1
SCHEMBL21444696 0.85 ALDH1A1 (0.53) ALDH1A1TACR1MAPK1L3MBTL1
SCHEMBL13108402 0.85 TACR1 (0.58) ALDH1A1TACR1
SCHEMBL2059140 0.85 TACR1 (0.58) ALDH1A1TACR1
SCHEMBL8348342 0.85 ALDH1A1 (0.53) ALDH1A1TACR1LMNASMN1; SMN2MAPK1
SCHEMBL28750936 0.84 TACR1 (0.61) ALDH1A1CASP1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025085756-A1 MACROCYCLIC COMPOUNDS AND METHODS OF TREATMENT UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2025-04-24 WO disclosed
US-10745692-B2 Production method for charged non-protein amino acid-containing peptide THE UNIVERSITY OF TOKYO (JP) 2020-08-18 US disclosed
US-20160289668-A1 Production Method for Charged Non-Protein Amino Acid-Containing Peptide THE UNIVERSITY OF TOKYO (JP) 2016-10-06 US disclosed
EP-3031915-A1 PRODUCTION METHOD FOR CHARGED NON-PROTEIN AMINO ACID-CONTAINING PEPTIDE The University of Tokyo (JP) 2016-06-15 EP disclosed
WO-2015019999-A1 PRODUCTION METHOD FOR CHARGED NON-PROTEIN AMINO ACID-CONTAINING PEPTIDE 国立大学法人東京大学 (JP) 2015-02-12 WO disclosed
US-8178490-B2 Polybasic bacterial efflux pump inhibitors and therapeutic uses thereof REMPEX PHARMACEUTICALS, INC. (US) 2012-05-15 US disclosed
US-20100152098-A1 POLYBASIC BACTERIAL EFFLUX PUMP INHIBITORS AND THERAPEUTIC USES THEREOF MPEX PHARMACEUTICALS, INC. (US) 2010-06-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100152098-A1 POLYBASIC BACTERIAL EFFLUX PUMP INHIBITORS AND THERAPEUTIC USES THEREOF ABCB11, ABCB1, SLC47A1 ALDH1A1 4062/4885CASP1 3606/4885HTT 3780/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.