SCHEMBL5019718

SCHEMBL5019718

CC1=C(c2cnc(NC(=O)c3cc(F)ccc3Cl)cn2)CN(c2nnn(C)n2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.36
ABL1 P00519 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
MAP3K5 Q99683 2/20 0.35
IL2 P60568 1/20 0.34
TP53 P04637 1/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34
P2RX7 Q99572 1/20 0.33
WNT1 P04628 1/20 0.33
DYRK1A Q13627 1/20 0.33
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33
STIM1 Q13586 1/20 0.33
ORAI1 Q96D31 1/20 0.33
ORAI2 Q96SN7 1/20 0.33
CYP2C19 P33261 1/20 0.33
RET P07949 1/20 0.33
PPARG P37231 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1780512 0.93 THRB (0.35) THRBABL1NPC1RAB9AMAP3K5
SCHEMBL3827961 0.90 HTR1F (0.42) NPC1RAB9AMAP3K5IL2TP53
SCHEMBL10819910 0.85 MAP3K5 (0.39) NPC1RAB9AMAP3K5IL2TP53
SCHEMBL5019623 0.85 PTPN11 (0.34) NPC1RAB9AMAP3K5IL2WNT1
SCHEMBL3826508 0.85 KMT2A (0.47) ABL1NPC1RAB9AMAP3K5TP53
SCHEMBL5019588 0.85 GRM5 (0.36) MAP3K5IL2KDM4EWNT1DYRK1A
SCHEMBL3824488 0.84 IL2 (0.42) IL2P2RX7STIM1ORAI1ORAI2
SCHEMBL5019579 0.84 KMT2A (0.39) NPC1RAB9AMAP3K5IL2TP53
SCHEMBL5019603 0.84 KMT2A (0.39) NPC1RAB9AMAP3K5IL2TP53
SCHEMBL5019754 0.84 GRM5 (0.40) THRBTP53LMNAIKBKBCHUK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064808-A1 TETRAZOLYL - TETRAHYDROPYRIDINE COMPOUNDS FOR INFLAMMATION AND IMMUNE - RELATED USES SYNTA PHARMACEUTICALS CORP (US) 2012-05-18 WO disclosed