SCHEMBL5019754

SCHEMBL5019754

CC1=C(c2ccc(NC(=O)c3cc(F)ccc3Cl)cc2)CN(c2nnn(C)n2)CC1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.40
NR3C1 P04150 1/20 0.39
NPY1R P25929 1/20 0.38
NPY2R P49146 1/20 0.38
THRB P10828 1/20 0.38
PTGES O14684 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
RECQL P46063 1/20 0.37
AVPR2 P30518 1/20 0.36
AVPR1A P37288 1/20 0.36
PPARG P37231 2/20 0.36
IKBKB O14920 2/20 0.36
CHUK O15111 1/20 0.36
PTPN11 Q06124 1/20 0.36
WDR5 P61964 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5019587 0.88 LCLAT1 (0.40) THRBMEN1KMT2ATP53
SCHEMBL1781784 0.88 SMO (0.44) MEN1KMT2ALMNAWDR5
SCHEMBL5019637 0.85 KMT2A (0.41) NR3C1MEN1KMT2ATP53WDR5
SCHEMBL5019716 0.84 RAB9A (0.47) MEN1KMT2ALMNATP53
SCHEMBL1781817 0.84 KMT2A (0.50) MEN1KMT2ALMNATP53
SCHEMBL1781495 0.84 RAB9A (0.38) NR3C1MEN1KMT2ATP53PTPN11
SCHEMBL5019718 0.84 THRB (0.36) THRBLMNATP53PPARGIKBKB
SCHEMBL5019717 0.83 CRACR2A (0.39)
SCHEMBL5019638 0.83 KMT2A (0.41) KMT2ALMNATP53AVPR2WDR5
SCHEMBL5019609 0.83 AVPR2 (0.42) MEN1KMT2ALMNATP53AVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064808-A1 TETRAZOLYL - TETRAHYDROPYRIDINE COMPOUNDS FOR INFLAMMATION AND IMMUNE - RELATED USES SYNTA PHARMACEUTICALS CORP (US) 2012-05-18 WO disclosed