SCHEMBL5019723

SCHEMBL5019723

CCC1=C(c2ccc(NC(=O)c3cccc(F)c3F)cc2)CN(c2nnn(C)n2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
AURKA O14965 2/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
CHRNA7 P36544 7/20 0.36
KCNH2 Q12809 7/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
MCL1 Q07820 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MEN1 O00255 2/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
LCLAT1 Q6UWP7 1/20 0.35
JAK1 P23458 1/20 0.35
WDR5 P61964 1/20 0.35
AURKB Q96GD4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5019601 0.92 SMN1; SMN2 (0.37) KMT2AAURKACTDSP1CHRNA7KCNH2
SCHEMBL5019681 0.91 SMN1; SMN2 (0.36) KMT2AAURKACTDSP1CHRNA7KCNH2
SCHEMBL5019638 0.89 KMT2A (0.41) KMT2AAURKACTDSP1CHRNA7KCNH2
SCHEMBL15356919 0.86 KMT2A (0.32) KMT2ATP53MAPTKDM4E
SCHEMBL5019751 0.83 RAB9A (0.38) KMT2AAURKACTDSP1CHRNA7KCNH2
SCHEMBL5019621 0.82 KDM4E (0.38) KMT2AAURKACTDSP1CHRNA7KCNH2
SCHEMBL5019609 0.82 AVPR2 (0.42) KMT2ACTDSP1CHRNA7KCNH2SMN1; SMN2
SCHEMBL1781817 0.82 KMT2A (0.50) KMT2ACTDSP1CHRNA7KCNH2SMN1; SMN2
SCHEMBL5019602 0.82 SMYD3 (0.36) SMN1; SMN2MAPTPOLB
SCHEMBL5019637 0.81 KMT2A (0.41) KMT2ACTDSP1CHRNA7KCNH2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064808-A1 TETRAZOLYL - TETRAHYDROPYRIDINE COMPOUNDS FOR INFLAMMATION AND IMMUNE - RELATED USES SYNTA PHARMACEUTICALS CORP (US) 2012-05-18 WO disclosed