SCHEMBL5020190

SCHEMBL5020190

CC(C)(NS(=O)(=O)c1ccc(-c2ccc(NC(=O)c3ccc(F)c(F)c3)cc2)cc1)C1CN=NN1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 2/20 0.48
KCNQ3 O43525 4/20 0.40
KCNQ2 O43526 4/20 0.40
HTR2B P41595 1/20 0.40
MAPT P10636 5/20 0.39
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALOX12 P18054 1/20 0.39
ATM Q13315 1/20 0.38
TP53 P04637 2/20 0.38
KCNE1 P15382 1/20 0.38
KCNQ1 P51787 1/20 0.38
BDKRB1 P46663 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
BCL9 O00512 1/20 0.38
CTNNB1 P35222 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5020144 0.88 PRMT1 (0.44) KCNQ3KCNQ2MAPTALDH1A1MEN1
SCHEMBL3078521 0.77 USP30 (0.49) USP30KCNQ3KCNQ2HTR2BMAPT
SCHEMBL3083418 0.75 KCNQ3 (0.44) USP30KCNQ3KCNQ2HTR2BMAPT
SCHEMBL14615719 0.72 GPR55 (0.59) USP30KCNQ3KCNQ2HTR2BMAPT
SCHEMBL3088538 0.70 MMP2 (0.67)
SCHEMBL5020143 0.69 MMP8 (0.39)
SCHEMBL14012554 0.69 MMP2 (0.60) HTR2BLMNA
SCHEMBL12855775 0.69 MMP2 (0.60) HTR2BLMNA
SCHEMBL5020184 0.68 BRD4 (0.43) MEN1KMT2A
SCHEMBL23352871 0.65 TRPV1 (0.68) KCNQ3KCNQ2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064943-A2 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed