SCHEMBL5023391

SCHEMBL5023391

C=C(C)NC(=O)c1c(F)cccc1F

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
CES2 O00748 2/20 0.48
CES1 P23141 2/20 0.48
PPIA P62937 1/20 0.46
JAK2 O60674 1/20 0.46
JAK1 P23458 1/20 0.46
TYK2 P29597 1/20 0.46
HTT P42858 1/20 0.46
NOD2 Q9HC29 1/20 0.46
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
GAA P10253 1/20 0.43
LMNA P02545 1/20 0.42
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5022120 0.85 ITGA4 (0.41) KMT2AMEN1CES2CES1TYK2
SCHEMBL13328951 0.84 CES2 (0.52) KMT2AMEN1CES2CES1PPIA
SCHEMBL31259499 0.83 CES2 (0.61) KMT2AMEN1CES2CES1PPIA
SCHEMBL8170361 0.81 MEN1 (0.49) KMT2AMEN1CES2CES1PPIA
SCHEMBL9363197 0.78 KMT2A (0.57) KMT2AMEN1CES2CES1PPIA
SCHEMBL11099551 0.78 CES2 (0.54) KMT2AMEN1CES2CES1PPIA
SCHEMBL27309508 0.77 KMT2A (0.55) KMT2AMEN1CES2CES1PPIA
SCHEMBL20387809 0.77 ALDH1A1 (0.50) PPIAJAK2JAK1TYK2RAB9A
SCHEMBL10572106 0.77 PPIA (0.54) KMT2AMEN1CES2CES1PPIA
SCHEMBL6989541 0.76 JAK2 (0.53) KMT2AMEN1CES2CES1PPIA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064744-A2 TETRAHYDROQUINOLINE AND RELATED BICYCLIC COMPOUNDS FOR INHIBITION OF RORϒ ACTIVITY AND THE TREATMENT OF DISEASE LYCERA CORPORATION (US) 2012-05-18 WO disclosed