SCHEMBL5023609

SCHEMBL5023609

COc1ccc(NC(=O)c2ccccc2Cl)cc1OC

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.72
KMT2A Q03164 5/20 0.70
ALDH1A1 P00352 5/20 0.70
KDM4E B2RXH2 3/20 0.70
MEN1 O00255 3/20 0.67
GRM4 Q14833 8/20 0.67
SMN1; SMN2 Q16637 5/20 0.66
MAPT P10636 5/20 0.66
NPC1 O15118 4/20 0.66
RAB9A P51151 4/20 0.66
HPGD P15428 1/20 0.66
HTT P42858 1/20 0.64
POLB P06746 2/20 0.64
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
CYP2D6 P10635 1/20 0.64
CYP2C9 P11712 1/20 0.64
CYP2C19 P33261 1/20 0.64
MAPK1 P28482 1/20 0.63
USP2 O75604 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL195970 0.91 SMN1; SMN2 (0.78) PTGS2KMT2AALDH1A1KDM4EMEN1
SCHEMBL11691716 0.88 ALDH1A1 (0.65) PTGS2KMT2AALDH1A1KDM4EMEN1
SCHEMBL11313551 0.88 KDM4E (0.62) PTGS2KMT2AALDH1A1KDM4EMEN1
SCHEMBL12181724 0.88 ALDH1A1 (0.65) PTGS2KMT2AALDH1A1KDM4EMEN1
SCHEMBL12189396 0.84 KMT2A (0.69) PTGS2KMT2AALDH1A1KDM4EMEN1
SCHEMBL23202525 0.83 KMT2A (0.67) PTGS2KMT2AALDH1A1KDM4EMEN1
SCHEMBL28568665 0.83 PTGS2 (0.55) PTGS2KMT2AALDH1A1KDM4EMEN1
SCHEMBL15164883 0.82 HTT (0.74) PTGS2KMT2AALDH1A1KDM4EMEN1
SCHEMBL10520535 0.82 METAP2 (0.68) PTGS2KMT2AALDH1A1KDM4EMEN1
SCHEMBL31078090 0.81 RORC (0.61) PTGS2KMT2AALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638556-B1 2-AMINOBENZOTHIAZOLES AS CB1 RECEPTOR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-04-02 EP claimed