SCHEMBL5025531

SCHEMBL5025531

CP(C)(=O)c1ccc(-c2nc3c(N)ncnc3[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 1/20 0.40
PI4K2B Q8TCG2 1/20 0.40
PI4K2A Q9BTU6 1/20 0.40
PI4KB Q9UBF8 1/20 0.40
PARP1 P09874 5/20 0.36
TNKS O95271 4/20 0.36
TNKS2 Q9H2K2 4/20 0.36
PRMT5 O14744 1/20 0.35
PIK3CG P48736 2/20 0.35
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADK P55263 2/20 0.34
RPS6KA3 P51812 1/20 0.34
MAP4K4 O95819 2/20 0.33
NUDT1 P36639 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29044196 0.78 ABL1 (0.47) PI4KAPI4K2BPI4K2API4KBPARP1
SCHEMBL9175737 0.77 PI4KA (0.64) PI4KAPI4K2BPI4K2API4KBPRMT5
SCHEMBL29459254 0.77 PI4KA (0.64) PI4KAPI4K2BPI4K2API4KBPRMT5
SCHEMBL15756441 0.77 MAP4K4 (0.48) PI4KAPI4K2BPI4K2API4KBPARP1
SCHEMBL15756646 0.77 ALDH1A1 (0.43) PI4KAPI4K2BPI4K2API4KBPARP1
SCHEMBL15756556 0.77 PIK3CD (0.50) PI4KAPI4K2BPI4K2API4KBPARP1
SCHEMBL15756483 0.68 PIK3CD (0.54) PI4K2APARP1TNKSTNKS2PIK3CG
Hydrochloric Acid SCHEMBL8595784 0.67 MAP4K4 (0.54) PI4KAPI4K2BPI4K2API4KBPARP1
SCHEMBL5025525 0.66 ADK (0.33) PARP1ADK
SCHEMBL8653515 0.65 PI4KA (0.42) PI4KAPI4K2BPI4K2API4KBPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940843-A2 UNSATURATED HETEROCYCLIC DERIVATIVES ARIAD PHARMACEUTICALS, INC. (US) 2008-07-09 EP disclosed
WO-2007021937-A2 UNSATURATED HETEROCYCLIC DERIVATIVES ARIAD PHARMACEUTICALS, INC. (US) 2007-02-22 WO disclosed