SCHEMBL5025525

SCHEMBL5025525

CP(C)(=O)c1ccc(-c2nc(N)c3nc[nH]c3n2)cc1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADK P55263 1/20 0.33
ADORA3 P0DMS8 1/20 0.31
ADORA1 P30542 1/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15756771 0.79 DPP4 (0.41) ADK
SCHEMBL1741363 0.78 ADORA2A (0.46) ADKADORA3ADORA1
SCHEMBL17815691 0.78 RIPK1 (0.44) PARP1
SCHEMBL15756598 0.76 ALDH1A1 (0.43) ADORA3ADORA1
SCHEMBL30747788 0.75 GDA (0.33)
SCHEMBL27249496 0.75 GDA (0.33)
SCHEMBL28084733 0.72 TLR9 (0.47) ADORA3ADORA1
SCHEMBL22019266 0.70 L3MBTL1 (0.37)
SCHEMBL11004734 0.69 LMNA (0.46) ADORA1
SCHEMBL7821784 0.69 ALDH1A1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940843-A2 UNSATURATED HETEROCYCLIC DERIVATIVES ARIAD PHARMACEUTICALS, INC. (US) 2008-07-09 EP disclosed
WO-2007021937-A2 UNSATURATED HETEROCYCLIC DERIVATIVES ARIAD PHARMACEUTICALS, INC. (US) 2007-02-22 WO disclosed