SCHEMBL5026434

SCHEMBL5026434

CC1(CCc2cccc(Br)c2)Cc2ccccc2C(NOC(=O)C(F)(F)F)=N1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 8/20 0.41
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 1/20 0.33
ORAI1 Q96D31 1/20 0.33
MTOR P42345 1/20 0.33
UTS2R Q9UKP6 1/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP2C9 P11712 1/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5028541 0.85 BACE1 (0.56) BACE1CYP1A2CYP2C19CYP2C9CYP3A4
Trifluoroacetic Acid SCHEMBL4995659 0.81 BACE1 (0.53) BACE1MEN1KMT2AORAI1TP53
SCHEMBL5030034 0.78 HCAR3 (0.35) MEN1KMT2AMAPTORAI1UTS2R
SCHEMBL5026581 0.77 MAPT (0.34) BACE1MEN1KMT2AMAPTORAI1
SCHEMBL8234637 0.76 BACE1 (0.43) BACE1
SCHEMBL5030127 0.71 BACE1 (0.36) BACE1KMT2AUTS2RCYP1A2CYP2D6
SCHEMBL5024092 0.69 NOS3 (0.41) MEN1KMT2AMAPT
SCHEMBL5024194 0.69 CYP1A2 (0.33) MEN1KMT2ACYP1A2CYP2D6CYP2C19
SCHEMBL5025605 0.68 MAPT (0.36) MEN1KMT2AMAPTORAI1CYP1A2
SCHEMBL18064339 0.68 TAAR1 (0.49) MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957462-A2 NOVEL 2-AMINO-HETEROCYCLES UDEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES Astra Zeneca AB (SE) 2008-08-20 EP claimed
WO-2007058583-A2 NOVEL 2-AMINO-HETEROCYCLES USEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES ASTRAZENECA AB (SE) 2007-05-24 WO claimed
EP-1957462-A2 NOVEL 2-AMINO-HETEROCYCLES UDEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES Astra Zeneca AB (SE) 2008-08-20 EP disclosed
WO-2007058583-A2 NOVEL 2-AMINO-HETEROCYCLES USEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES ASTRAZENECA AB (SE) 2007-05-24 WO disclosed