SCHEMBL5028952

SCHEMBL5028952

COc1ccc(C2CN(C(C)=S)CCO2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
MAPT P10636 3/20 0.44
HPGD P15428 2/20 0.44
GAA P10253 2/20 0.44
APOBEC3G Q9HC16 1/20 0.44
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
FKBP1A P62942 2/20 0.41
POLB P06746 1/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
PDE2A O00408 1/20 0.40
CYP2D6 P10635 1/20 0.40
GSK3B P49841 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19049385 0.86 PDE2A (0.44) ALDH1A1MAPTHPGDGAAL3MBTL1
SCHEMBL6243985 0.84 CNR2 (0.42) PDE2ACNR2
SCHEMBL21438214 0.84 CYP2D6 (0.44) KMT2AMEN1L3MBTL1SMN1; SMN2LMNA
SCHEMBL6444671 0.84 CNR2 (0.44) ALDH1A1HPGDKMT2AMEN1PDE2A
SCHEMBL5028958 0.83 ALDH1A1 (0.43) ALDH1A1HPGDPOLBPDE2A
SCHEMBL21438238 0.81 PDE2A (0.39) ALDH1A1MAPTHPGDGAAAPOBEC3G
SCHEMBL19002801 0.80 MMP1 (0.45) ALDH1A1MAPTGAAKMT2AL3MBTL1
SCHEMBL19002794 0.80 DRD3 (0.47) ALDH1A1HPGDGAASMN1; SMN2FKBP1A
SCHEMBL5029162 0.78 AKR1C3 (0.41)
SCHEMBL24394579 0.78 CYP2D6 (0.46) CYP2D6GSK3BCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007393-A2 THIAZOLE AND THIOPHENE ANALOGUES, AND THEIR USE IN TREATING AUTOIMMUNE DISEASES AND CANCERS Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College (US) 2008-12-31 EP disclosed
WO-2007118149-A2 THIAZOLE AND THIOPHENE ANALOGUES, AND THEIR USE IN TREATING AUTOIMMUNE DISEASES AND CANCERS BOARD OF SUPERVISORS OF LOUISIANA STATE UNIVERSITY AND AGRICULTURAL AND MECHANICAL LOLLEGE (US) 2007-10-18 WO disclosed