SCHEMBL5030309

SCHEMBL5030309

c1ccc(-c2ccccc2-c2ccc3c(c2)c2cc(-c4ccccc4-c4ccccn4)ccc2n3-c2ccc3oc4ccc(-n5c6ccc(-c7ccccc7-c7ccccn7)cc6c6cc(-c7ccccc7-c7ccccn7)ccc65)cc4c3c2)nc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 3/20 0.36
GRM5 P41594 4/20 0.35
MAPK14 Q16539 1/20 0.35
PIM1 P11309 1/20 0.34
PIM3 Q86V86 1/20 0.34
DHFR P00374 2/20 0.33
NPY5R Q15761 1/20 0.33
NPC1 O15118 3/20 0.33
MAPT P10636 1/20 0.33
AHR P35869 1/20 0.32
PRKDC P78527 1/20 0.32
HSD17B10 Q99714 3/20 0.32
TP53 P04637 2/20 0.32
RAB9A P51151 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
PKM P14618 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12114616 1.00 TGFBR1 (0.36) TGFBR1GRM5MAPK14PIM1PIM3
SCHEMBL5028244 0.97 GRM5 (0.40) TGFBR1GRM5MAPK14PIM1PIM3
SCHEMBL13471349 0.97 TGFBR1 (0.34) TGFBR1GRM5MAPK14PIM1PIM3
SCHEMBL11946077 0.97 NPY5R (0.37) TGFBR1GRM5MAPK14PIM1PIM3
SCHEMBL13471317 0.97 NPC1 (0.38) TGFBR1GRM5MAPK14PIM1PIM3
SCHEMBL10123521 0.97 NPY5R (0.37) TGFBR1GRM5MAPK14PIM1PIM3
SCHEMBL13471340 0.96 GRM5 (0.37) TGFBR1GRM5MAPK14PIM1PIM3
SCHEMBL20097822 0.94 NPY5R (0.36) TGFBR1GRM5MAPK14PIM1PIM3
SCHEMBL13471347 0.94 NPY5R (0.36) TGFBR1GRM5MAPK14PIM1PIM3
SCHEMBL16451563 0.94 GRM5 (0.38) TGFBR1GRM5MAPK14PIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 303 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11765967-B2 Highly efficient OLED devices with very short decay times UDC IRELAND LIMITED (IE) 2023-09-19 US disclosed
US-11765967-B2 Highly efficient OLED devices with very short decay times UDC IRELAND LIMITED (IE) 2023-09-19 US disclosed
EP-4060757-A1 HIGHLY EFFICIENT OLED DEVICES WITH VERY SHORT DECAY TIMES UDC Ireland Limited (IE) 2022-09-21 EP disclosed
US-20220199934-A1 LUMINESCENT FILM, ORGANIC ELECTROLUMINESCENT ELEMENT, ORGANIC MATERIAL COMPOSITION AND METHOD FOR PRODUCING ORGANIC ELECTROLUMINESCENT ELEMENT UDC IRELAND LIMITED (IE) 2022-06-23 US disclosed
US-20220149300-A1 HIGHLY EFFICIENT OLED DEVICES WITH VERY SHORT DECAY TIMES UDC IRELAND LTD (IE) 2022-05-12 US disclosed
EP-3356369-B1 BENZIMIDAZOLO[1,2-A]BENZIMIDAZOLE CARRYING TRIAZINE GROUPS FOR ORGANIC LIGHT EMITTING DIODES IDEMITSU KOSAN CO (JP) 2022-05-04 EP disclosed
EP-3304612-B1 HIGHLY EFFICIENT OLED DEVICES WITH VERY SHORT DECAY TIMES UDC IRELAND LTD (IE) 2022-05-04 EP disclosed
US-11302882-B2 Luminescent film, organic electroluminescent element, organic material composition and method for producing organic electroluminescent element MERCK PATENT GMBH (DE) 2022-04-12 US disclosed
US-11174258-B2 Benzimidazolo[1,2-a]benzimidazole derivatives for organic light emitting diodes IDEMITSU KOSAN CO., LTD. (JP) 2021-11-16 US disclosed
EP-3126371-B1 METAL COMPLEXES, COMPRISING CARBENE LIGANDS HAVING AN O-SUBSTITUTED NON-CYCLOMETALATED ARYL GROUP AND THEIR USE IN ORGANIC LIGHT EMITTING DIODES UDC IRELAND LTD (IE) 2021-11-10 EP disclosed
US-20120037889-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT, DISPLAY DEVICE AND ILLUMINATION DEVICE KONICA MINOLTA HOLDINGS, INC. (JP) 2012-02-16 US disclosed
US-20120018714-A1 ORGANIC ELECTROLUMINESCENT DEVICE, DISPLAY APPARATUS, AND LIGHTING APPARATUS KONICA MINOLTA HOLDINGS, INC. (JP) 2012-01-26 US disclosed
US-20120018714-A1 ORGANIC ELECTROLUMINESCENT DEVICE, DISPLAY APPARATUS, AND LIGHTING APPARATUS KONICA MINOLTA HOLDINGS, INC. (JP) 2012-01-26 US disclosed
US-20120007072-A1 ORGANIC ELECTROLUMINESCENT ELEMENT MERCK PATENT GMBH (DE) 2012-01-12 US disclosed
US-20120007072-A1 ORGANIC ELECTROLUMINESCENT ELEMENT MERCK PATENT GMBH (DE) 2012-01-12 US disclosed
US-20110260152-A1 ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE, AND ILLUMINATION DEVICE KONICA MINOLTA HOLDINGS, INC. (JP) 2011-10-27 US disclosed
US-20110260152-A1 ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE, AND ILLUMINATION DEVICE KONICA MINOLTA HOLDINGS, INC. (JP) 2011-10-27 US disclosed
US-20110006670-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT, NEW COMPOUND FOR THE SAME, DISPLAY DEVICE AND LIGHTING DEVICE USING THE SAME KONICA MINOLTA HOLDINGS, INC. (JP) 2011-01-13 US disclosed
US-20110006670-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT, NEW COMPOUND FOR THE SAME, DISPLAY DEVICE AND LIGHTING DEVICE USING THE SAME KONICA MINOLTA HOLDINGS, INC. (JP) 2011-01-13 US disclosed
US-20090284138-A1 ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE AND LIGHTING DEVICE KONICA MINOLTA HOLDINGS, INC. (JP) 2009-11-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11174258-B2 Benzimidazolo[1,2-a]benzimidazole derivatives for organic light emitting diodes KCNH2, KCNH3, KCNJ2 TGFBR1 155/4885GRM5 3032/4885MAPK14 4106/4885
US-20110006670-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT, NEW COMPOUND FOR THE SAME, DISPLAY DEVICE AND LIGHTING DEVICE USING THE SAME AOC2, AOC3, CDYL TGFBR1 2661/4885GRM5 2093/4885MAPK14 3907/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.