SCHEMBL5032170

SCHEMBL5032170

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nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
TDP1 Q9NUW8 1/20 0.55
USP2 O75604 1/20 0.43
SLCO1B1 Q9Y6L6 1/20 0.43
KDM4E B2RXH2 2/20 0.41
PDE4A P27815 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1129672 1.00 LMNA (0.58) LMNAL3MBTL1TDP1USP2SLCO1B1
SCHEMBL1671960 1.00 LMNA (0.58) LMNAL3MBTL1TDP1USP2SLCO1B1
Mannitol SCHEMBL4971188 1.00 LMNA (0.58) LMNAL3MBTL1TDP1USP2SLCO1B1
SCHEMBL6542053 0.97 TDP1 (0.60) LMNAL3MBTL1TDP1USP2SLCO1B1
SCHEMBL11423256 0.97 TDP1 (0.60) LMNAL3MBTL1TDP1USP2SLCO1B1
SCHEMBL8075862 0.97 TDP1 (0.60) LMNAL3MBTL1TDP1USP2SLCO1B1
SCHEMBL6541711 0.95 LMNA (0.50) LMNAL3MBTL1TDP1USP2SLCO1B1
SCHEMBL15892815 0.93 LMNA (0.50) LMNAL3MBTL1TDP1USP2SLCO1B1
SCHEMBL14654998 0.89 LMNA (0.37) LMNAL3MBTL1TDP1
Succinic Acid SCHEMBL5075718 0.85 USP2 (0.47) LMNAL3MBTL1TDP1USP2SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9907854-B2 Crosslinking reagents, macromolecules, therapeutic bioconjugates, and synthetic methods thereof CellMosaic, Inc. (US) 2018-03-06 US disclosed
US-9907854-B2 Crosslinking reagents, macromolecules, therapeutic bioconjugates, and synthetic methods thereof CellMosaic, Inc. (US) 2018-03-06 US disclosed
US-20170065726-A1 NOVEL CROSSLINKING REAGENTS, MACROMOLECULES, THERAPEUTIC BIOCONJUGATES, AND SYNTHETIC METHODS THEREOF CELLMOSAIC INC (US) 2017-03-09 US disclosed
US-20170065726-A1 NOVEL CROSSLINKING REAGENTS, MACROMOLECULES, THERAPEUTIC BIOCONJUGATES, AND SYNTHETIC METHODS THEREOF CELLMOSAIC INC (US) 2017-03-09 US disclosed
US-9511150-B2 Crosslinking reagents, macromolecules, therapeutic bioconjugates, and synthetic methods thereof CellMosaic, Inc. (US) 2016-12-06 US disclosed
US-8907079-B2 Crosslinking reagents, macromolecules, therapeutic conjugates, and synthetic methods thereof CELLMOSAIC INC. (US) 2014-12-09 US disclosed
US-20140206903-A1 NOVELCROSSLINKING REAGENTS, MACROMOLECULES, THERAPEUTIC CONJUGATES, AND SYNTHETIC METHODS THEREOF CELLMOSAIC INC (US) 2014-07-24 US disclosed
CN-103476932-A Nucleic acid modulators of CLEC-2 REGADO BIOSCIENCES INC 2013-12-25 CN disclosed
WO-2008141799-A1 OLIGOPHOSPHORAMIDATES ROCHE DIAGNOSTICS GMBH (DE) 2008-11-27 WO disclosed
US-6274115-B1 PROVIDING MICELLULAR PARTICLES COMPRISING PHOSPHOLIPID MOLECULES WHICH ARE STABLE TO LEAKAGE IN VITRO AND IN VIVO; MODIFYING MICELLULAR PARTILCES; INTRODUCING INTO BLOOD STREAM; INCORPORATINGAGENT FOR DIAGNOSIS OR THERAPY INTO SECND GROUP GILEAD SCIENCES, INC. 2001-08-14 US disclosed
US-5441745-A Marking tumors in the body; biodegradable VESTAR, INC. (US) 1995-08-15 US disclosed
US-5435989-A Tumors, phospholipid micelles VESTAR, INC. (US) 1995-07-25 US disclosed
EP-0182131-B1 THE USE OF MICELLULAR PARTICLE FOR MAKING COMPOSITIONS FOR TARGETING TUMORS IN HUMANS VESTAR, INC. (US) 1991-12-18 EP disclosed
EP-0179444-B1 USE OF A MICELLULAR PARTICLE COMPOSITION ENCAPSULATING A CHEMOTHERAPEUTIC AGENT FOR INTRAVENOUS TARGETING TO TUMORS VESTAR, INC. (US) 1991-06-12 EP disclosed
US-5019369-A Method of targeting tumors in humans VESTAR, INC. (US) 1991-05-28 US disclosed
EP-0182131-A1 The use of micellular particle for making compositions for targeting tumors in humans VESTAR, INC. (US) 1986-05-28 EP disclosed
EP-0179444-A2 Use of a micellular particle composition encapsulating a chemotherapeutic agent for intravenous targeting to tumors VESTAR, INC. (US) 1986-04-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170065726-A1 NOVEL CROSSLINKING REAGENTS, MACROMOLECULES, THERAPEUTIC BIOCONJUGATES, AND SYNTHETIC METHODS THEREOF CD44, ADH1C, EPCAM LMNA 4262/4885L3MBTL1 2520/4885TDP1 4207/4885
US-20140206903-A1 NOVELCROSSLINKING REAGENTS, MACROMOLECULES, THERAPEUTIC CONJUGATES, AND SYNTHETIC METHODS THEREOF CD44, ADH1C, EPCAM LMNA 4454/4885L3MBTL1 2862/4885TDP1 4314/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.