SCHEMBL5034461

SCHEMBL5034461

CCNC(=O)CCCN[C@@H](CC)C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FAAH O00519 5/20 0.46
CAPN1 P07384 4/20 0.42
NOD1 Q9Y239 2/20 0.37
EPHX2 P34913 1/20 0.35
CAPN2 P17655 1/20 0.34
ALB P02768 1/20 0.34
CASP2 P42575 1/20 0.33
DNM1 Q05193 2/20 0.33
TSHR P16473 2/20 0.33
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14186683 0.87 NOD1 (0.47) FAAHNOD1EPHX2CASP2DNM1
SCHEMBL5037670 0.87 NOD1 (0.47) FAAHNOD1EPHX2CASP2DNM1
SCHEMBL5038748 0.84 CA1 (0.35) FAAHNOD1TSHR
SCHEMBL6018656 0.81 CYP3A4 (0.51)
SCHEMBL10521386 0.81 AKR1B1 (0.39) TSHR
SCHEMBL2704035 0.81 AKR1B1 (0.39) TSHR
SCHEMBL14367747 0.81 PAOX (0.38) NOD1
SCHEMBL2704033 0.81 AKR1B1 (0.39) TSHR
SCHEMBL5038713 0.79 GAA (0.57) FAAHEPHX2
SCHEMBL562999 0.78 TSHR (0.47) EPHX2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339669-B1 N-ALKYLATED GABA COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS UCB PHARMA SA (BE) 2008-06-04 EP disclosed
US-7112612-B2 N-alkylated GABA compounds, processes for their preparation and their use as medicaments UCB S.A. (BE) 2006-09-26 US disclosed