SCHEMBL5034494

SCHEMBL5034494

CCCOc1ccc(C(=O)NCc2cccc(CC3(C(=O)O)C=CCO3)c2)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
TP53 P04637 2/20 0.41
NPC1 O15118 3/20 0.41
MAPT P10636 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ROCK2 O75116 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
ROCK1 Q13464 1/20 0.40
ESR1 P03372 1/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PTGIR P43119 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032948 0.93 ALDH1A1 (0.43) ALDH1A1TP53NPC1SMN1; SMN2RAB9A
SCHEMBL5029832 0.88 ALDH1A1 (0.39) ALDH1A1TP53NPC1MAPTSMN1; SMN2
SCHEMBL5031737 0.86 PPARA (0.41) PPARGPPARDPPARA
SCHEMBL5032956 0.85 HRH3 (0.38) ALDH1A1NPC1SMN1; SMN2RAB9AMEN1
SCHEMBL5031870 0.85 LMNA (0.43) ALDH1A1NPC1SMN1; SMN2RAB9AMEN1
SCHEMBL5030063 0.83 CHRM3 (0.42) ALDH1A1NPC1RAB9AESR1POLB
SCHEMBL5029835 0.82 ALDH1A1 (0.42) ALDH1A1TP53NPC1MAPTSMN1; SMN2
SCHEMBL5032820 0.80 PPARA (0.40) ALDH1A1NPC1PPARGPPARDPPARA
SCHEMBL5034466 0.77 HTT (0.43) ALDH1A1MAPTKMT2ALMNAPPARG
SCHEMBL3413951 0.75 PTPN11 (0.51) ALDH1A1TP53NPC1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7371777-B2 Cyclic compound and PPAR agonist EISAI CO., LTD. (JP) 2008-05-13 US disclosed
US-7371777-B2 Cyclic compound and PPAR agonist EISAI CO., LTD. (JP) 2008-05-13 US disclosed
US-7371777-B2 Cyclic compound and PPAR agonist EISAI CO., LTD. (JP) 2008-05-13 US disclosed