SCHEMBL5032948

SCHEMBL5032948

CCOc1ccc(C(=O)NCc2cccc(CC3(C(=O)O)C=CCO3)c2)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
NPC1 O15118 2/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
POLB P06746 3/20 0.42
TP53 P04637 2/20 0.40
ROCK1 Q13464 2/20 0.39
ROCK2 O75116 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ESR1 P03372 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HPGD P15428 1/20 0.38
FADS1 O60427 1/20 0.38
LMNA P02545 1/20 0.38
PTGIR P43119 1/20 0.38
PPARG P37231 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5034494 0.93 ALDH1A1 (0.42) ALDH1A1NPC1KMT2AMEN1RAB9A
SCHEMBL5029832 0.90 ALDH1A1 (0.39) ALDH1A1NPC1KMT2AMEN1RAB9A
SCHEMBL5032956 0.86 HRH3 (0.38) ALDH1A1NPC1KMT2AMEN1RAB9A
SCHEMBL5031870 0.86 LMNA (0.43) ALDH1A1NPC1KMT2AMEN1RAB9A
SCHEMBL5032820 0.86 PPARA (0.40) ALDH1A1NPC1HPGDPPARGPPARD
SCHEMBL5030063 0.84 CHRM3 (0.42) ALDH1A1NPC1RAB9APOLBESR1
SCHEMBL5032927 0.81 ALDH1A1 (0.43) ALDH1A1NPC1KMT2AMEN1RAB9A
SCHEMBL5031737 0.80 PPARA (0.41) PPARGPPARDPPARA
SCHEMBL5034466 0.79 HTT (0.43) ALDH1A1KMT2AHPGDLMNAPPARG
SCHEMBL5032738 0.76 PPARA (0.40) ALDH1A1HPGDLMNAPPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7371777-B2 Cyclic compound and PPAR agonist EISAI CO., LTD. (JP) 2008-05-13 US disclosed
US-7371777-B2 Cyclic compound and PPAR agonist EISAI CO., LTD. (JP) 2008-05-13 US disclosed
US-7371777-B2 Cyclic compound and PPAR agonist EISAI CO., LTD. (JP) 2008-05-13 US disclosed