SCHEMBL5034651

SCHEMBL5034651

CC(=O)Oc1c(C)cc(Cc2cc(C)c(O)c(C)c2)cc1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGB1 P09429 1/20 0.51
CXCL12 P48061 1/20 0.51
HTT P42858 2/20 0.46
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46
TP53 P04637 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
SHBG P04278 1/20 0.46
CFD P00746 1/20 0.39
PREP P48147 3/20 0.39
CELA1 Q9UNI1 2/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
POLB P06746 1/20 0.37
ESR1 P03372 3/20 0.37
ESR2 Q92731 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12445342 0.86 ALDH1A1 (0.44) HMGB1CXCL12HTTKDM4EHSD17B10
SCHEMBL12521523 0.83 CA1 (0.56) HTTKDM4EHSD17B10TP53GAA
SCHEMBL18567239 0.81 HTT (0.40) HMGB1CXCL12HTTKDM4EHSD17B10
SCHEMBL1979635 0.79 CYP4F2 (0.51) HTTKDM4EHSD17B10TP53GAA
SCHEMBL15443903 0.79 HSD17B10 (0.46) HTTKDM4EHSD17B10TP53GAA
SCHEMBL68876 0.78 SHBG (0.67) HMGB1CXCL12KDM4EGAAMAPT
SCHEMBL24202214 0.78 HTT (0.45) HTTKDM4EHSD17B10TP53GAA
SCHEMBL1974691 0.78 HTT (0.45) HTTKDM4EHSD17B10TP53GAA
SCHEMBL14137288 0.78 MAPT (0.48) HMGB1CXCL12GAAMAPTSHBG
SCHEMBL15443899 0.77 HTT (0.45) HTTKDM4EHSD17B10TP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9811008-B2 Image forming method, process cartridge, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2017-11-07 US disclosed
US-9766561-B2 Electrophotographic photosensitive member, process cartridge and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2017-09-19 US disclosed
EP-2633370-B1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KK (JP) 2017-04-26 EP disclosed
US-9557660-B2 Electrophotographic photosensitive member, process cartridge, electrophotographic apparatus, charge transport layer forming coating liquid, and method for manufacturing electrophotographic photosensitive member CANON KABUSHIKI KAISHA (JP) 2017-01-31 US disclosed
US-20170010556-A1 IMAGE FORMING METHOD, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2017-01-12 US disclosed
US-9529284-B2 Process cartridge, image forming method, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2016-12-27 US disclosed
US-20160291488-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2016-10-06 US disclosed
US-20160252831-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, ELECTROPHOTOGRAPHIC APPARATUS, CHARGE TRANSPORT LAYER FORMING COATING LIQUID, AND METHOD FOR MANUFACTURING ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER CANON KK (JP) 2016-09-01 US disclosed
US-9411307-B2 Process cartridge and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2016-08-09 US disclosed
US-9389522-B2 Electrophotographic photosensitive member, process cartridge, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2016-07-12 US disclosed
US-20130236823-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, ELECTROPHOTOGRAPHIC APPARATUS, AND METHOD OF MANUFACTURING ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER CANON KABUSHIKI KAISHA (JP) 2013-09-12 US disclosed
US-20130202326-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, ELECTROPHOTOGRAPHIC APPARATUS, AND METHOD OF MANUFACTURING ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER CANON KABUSHIKI KAISHA (JP) 2013-08-08 US disclosed
US-20130202327-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2013-08-08 US disclosed
US-20130029266-A1 METHOD FOR PRODUCING ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER CANON KABUSHIKI KAISHA (JP) 2013-01-31 US disclosed
US-20130029256-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2013-01-31 US disclosed
US-20120243904-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2012-09-27 US disclosed
WO-2012074082-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, ELECTROPHOTOGRAPHIC APPARATUS, AND METHOD OF MANUFACTURING ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER CANON KABUSHIKI KAISHA (JP) 2012-06-07 WO disclosed
WO-2012057349-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, ELECTROPHOTOGRAPHIC APPARATUS, AND METHOD OF MANUFACTURING ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER CANON KABUSHIKI KAISHA (JP) 2012-05-03 WO disclosed
WO-2012057350-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2012-05-03 WO disclosed
US-20110177438-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2011-07-21 US disclosed