SCHEMBL5034997

SCHEMBL5034997

CC(C)(CO)NS(=O)(=O)c1ccc(Cl)c(NC(=O)Oc2cnn3c(C(F)F)cc(-c4ccc(C(F)(F)F)cc4)nc23)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
POLB P06746 3/20 0.41
TP53 P04637 3/20 0.41
ALDH1A1 P00352 4/20 0.40
KMT2A Q03164 4/20 0.40
MAPT P10636 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
HTT P42858 1/20 0.39
LMNA P02545 1/20 0.38
MEN1 O00255 1/20 0.38
MAPK1 P28482 1/20 0.38
KIF18A Q8NI77 1/20 0.37
HPGD P15428 1/20 0.37
GLA P06280 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032676 0.93 ALDH1A1 (0.45) KDM4EPOLBTP53ALDH1A1KMT2A
SCHEMBL5041458 0.91 ALDH1A1 (0.40) KDM4EPOLBALDH1A1KMT2AMAPT
SCHEMBL5045903 0.89 POLB (0.51) KDM4EPOLBTP53ALDH1A1KMT2A
SCHEMBL5039141 0.88 KDM4E (0.49) KDM4EPOLBTP53ALDH1A1KMT2A
SCHEMBL5035029 0.87 TP53 (0.41) KDM4EPOLBTP53ALDH1A1KMT2A
SCHEMBL1938878 0.87 MAPT (0.39) KDM4EPOLBTP53ALDH1A1KMT2A
SCHEMBL1941032 0.85 KMT2A (0.40) KDM4EPOLBTP53ALDH1A1KMT2A
SCHEMBL5034987 0.83 KDM4E (0.41) KDM4EPOLBALDH1A1KMT2AMAPT
SCHEMBL1940323 0.83 MAPT (0.40) KDM4EPOLBTP53ALDH1A1KMT2A
SCHEMBL5039082 0.83 KDM4E (0.49) KDM4EPOLBTP53ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed