SCHEMBL5032676

SCHEMBL5032676

Cc1ccc(S(=O)(=O)NC(C)(C)CO)cc1NC(=O)Oc1cnn2c(C(F)F)cc(-c3ccc(C(F)(F)F)cc3)nc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
KDM4E B2RXH2 3/20 0.45
POLB P06746 3/20 0.43
TP53 P04637 2/20 0.43
KMT2A Q03164 4/20 0.42
MAPT P10636 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MEN1 O00255 2/20 0.40
LMNA P02545 2/20 0.39
HTT P42858 2/20 0.38
KIF18A Q8NI77 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MAPK1 P28482 1/20 0.37
USP2 O75604 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5034997 0.93 KDM4E (0.41) ALDH1A1KDM4EPOLBTP53KMT2A
SCHEMBL5034987 0.91 KDM4E (0.41) ALDH1A1KDM4EPOLBKMT2AMAPT
SCHEMBL5041096 0.89 POLB (0.56) ALDH1A1KDM4EPOLBTP53KMT2A
SCHEMBL5039141 0.88 KDM4E (0.49) ALDH1A1KDM4EPOLBTP53KMT2A
SCHEMBL5039334 0.88 ALDH1A1 (0.47) ALDH1A1KDM4EPOLBTP53KMT2A
SCHEMBL5035231 0.88 KIF18A (0.35) ALDH1A1KDM4EPOLBTP53KMT2A
SCHEMBL1941032 0.87 KMT2A (0.40) ALDH1A1KDM4EPOLBTP53KMT2A
SCHEMBL1938878 0.85 MAPT (0.39) ALDH1A1KDM4EPOLBTP53KMT2A
SCHEMBL1938936 0.84 ALDH1A1 (0.39) ALDH1A1KDM4EPOLBTP53KMT2A
SCHEMBL1940323 0.84 MAPT (0.40) ALDH1A1KDM4EPOLBTP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed