SCHEMBL503793

SCHEMBL503793

Ic1cnc(N2CCN3CCC2CC3)nc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 6/20 0.40
HTR3A P46098 5/20 0.40
KCNH2 Q12809 4/20 0.40
CHRNA1 P02708 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL503831 0.87 CHRNA1 (0.34) CHRNA7HTR3AKCNH2CHRNA1CHRNB2
SCHEMBL504169 0.82 HTR3A (0.52) CHRNA7HTR3AKCNH2
SCHEMBL235246 0.82 HTR3A (0.52) CHRNA7HTR3AKCNH2
SCHEMBL242574 0.82 CHRNA7 (0.40) CHRNA7HTR3AKCNH2
Hydrochloric Acid SCHEMBL3756715 0.81 CHRNA7 (0.40) CHRNA7HTR3AKCNH2
SCHEMBL244511 0.76 MAPT (0.40) CHRNA7HTR3AKCNH2
SCHEMBL1782928 0.72 FURIN (0.35) CHRNA7HTR3AKCNH2
SCHEMBL2900861 0.72 CHRNA7 (0.47) CHRNA7HTR3AKCNH2
SCHEMBL2899831 0.72 CYP2A6 (0.39) CHRNA7HTR3A
Fumaric Acid SCHEMBL503796 0.71 KCNH2 (0.43) CHRNA7HTR3AKCNH2CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120028967-A1 NOVEL DIAZA-BICYCLONONYL-PYRIMIDINYL DERIVATIVES AND THEIR MEDICAL USE NEUROSEARCH A/S (DK) 2012-02-02 US claimed
US-20120028967-A1 NOVEL DIAZA-BICYCLONONYL-PYRIMIDINYL DERIVATIVES AND THEIR MEDICAL USE NEUROSEARCH A/S (DK) 2012-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120028967-A1 NOVEL DIAZA-BICYCLONONYL-PYRIMIDINYL DERIVATIVES AND THEIR MEDICAL USE CHRNA5, CHRNA6, CHRNA3 CHRNA7 6/4885HTR3A 104/4885KCNH2 801/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.