SCHEMBL5039367

SCHEMBL5039367

CCN(CCN(C)C)C(=O)Oc1csc(N(C(=O)c2ccccc2Cl)c2ccc(Cl)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HTT P42858 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TP53 P04637 1/20 0.36
CYP11B1 P15538 1/20 0.35
UTS2R Q9UKP6 4/20 0.34
POLB P06746 2/20 0.34
TSPO P30536 2/20 0.34
CYP3A4 P08684 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
RAD52 P43351 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
DHODH Q02127 1/20 0.33
S1PR1 P21453 1/20 0.33
CFTR P13569 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5036024 0.94 ALDH1A1 (0.37) KDM4EALDH1A1HTTNPSR1MAPT
SCHEMBL5035235 0.91 CYP3A4 (0.45) ALDH1A1HTTNPSR1MAPTRAB9A
SCHEMBL5032571 0.91 KDM4E (0.42) KDM4EALDH1A1HTTNPSR1MAPT
SCHEMBL5032555 0.86 ALDH1A1 (0.44) KDM4EALDH1A1HTTNPSR1MAPT
SCHEMBL5039136 0.85 CYP3A4 (0.44) ALDH1A1HTTRAB9ASMN1; SMN2CYP11B1
SCHEMBL5041385 0.85 CYP3A4 (0.46) ALDH1A1HTTMAPTRAB9ASMN1; SMN2
SCHEMBL5032567 0.84 CYP3A4 (0.49) ALDH1A1NPSR1MAPTRAB9ASMN1; SMN2
SCHEMBL5035010 0.83 CYP3A4 (0.39) ALDH1A1HTTNPSR1MAPTRAB9A
SCHEMBL5036077 0.82 CYP3A4 (0.42) KDM4EALDH1A1HTTNPSR1MAPT
SCHEMBL5035132 0.81 KDM4E (0.45) KDM4EALDH1A1HTTNPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694673-B1 THIAZOLE DERIVATES HOFFMANN LA ROCHE (CH) 2008-01-16 EP claimed