SCHEMBL5041907

SCHEMBL5041907

O=C(O)c1cc(S(=O)(=O)C2CC2)ccc1OC1CCCC1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4C Q08493 2/20 0.42
PDE4D Q08499 2/20 0.42
FABP4 P15090 2/20 0.42
FABP5 Q01469 2/20 0.42
APEX1 P27695 1/20 0.42
MRGPRX1 Q96LB2 1/20 0.40
LNPEP Q9UIQ6 1/20 0.40
MAOB P27338 1/20 0.40
SLC6A9 P48067 2/20 0.39
SYK P43405 2/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
GRIK1 P39086 1/20 0.38
GRIA2 P42262 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5037977 0.97 APEX1 (0.42) PDE4APDE4BPDE4CPDE4DFABP4
SCHEMBL1811462 0.85 SLC6A9 (0.51) PDE4APDE4BPDE4CPDE4DFABP4
SCHEMBL2826409 0.84 SLC6A9 (0.52) PDE4APDE4BPDE4CPDE4DFABP4
SCHEMBL2824807 0.82 SLC6A9 (0.51) PDE4APDE4BPDE4CPDE4DAPEX1
SCHEMBL2825503 0.82 FABP4 (0.45) PDE4APDE4BPDE4CPDE4DFABP4
SCHEMBL5045483 0.79 FABP4 (0.43) PDE4APDE4BPDE4CPDE4DFABP4
SCHEMBL4422191 0.78 APEX1 (0.44) APEX1MRGPRX1SLC6A9
SCHEMBL5043956 0.77 SLC6A9 (0.45) PDE4APDE4BPDE4CPDE4DFABP4
SCHEMBL8962289 0.77 GAA (0.47) APEX1GAAKMT2A
SCHEMBL4424161 0.76 SLC6A9 (0.53) PDE4APDE4BPDE4CPDE4DAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656361-B1 PIPERAZINE WITH OR-SUBSTITUTED PHENYL GROUP AND THEIR USE AS GLYT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed