SCHEMBL5043956

SCHEMBL5043956

O=C(O)c1cc(S(=O)(=O)C2CC2)ccc1OCC1CC1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 5/20 0.45
S1PR3 Q99500 1/20 0.44
PIM1 P11309 1/20 0.41
PIM2 Q9P1W9 1/20 0.41
MRGPRX1 Q96LB2 1/20 0.41
APEX1 P27695 1/20 0.41
KCNH2 Q12809 2/20 0.41
SYK P43405 1/20 0.41
KMO O15229 2/20 0.40
FABP4 P15090 1/20 0.39
FABP5 Q01469 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
BRD4 O60885 1/20 0.38
KAT6A Q92794 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2824930 0.85 SLC6A9 (0.59) SLC6A9S1PR3KCNH2BRD4
SCHEMBL5045383 0.82 BRD4 (0.48) SLC6A9S1PR3APEX1KCNH2SYK
SCHEMBL5043166 0.82 S1PR3 (0.45) SLC6A9S1PR3APEX1KCNH2SYK
SCHEMBL1813202 0.81 SLC6A9 (0.54) SLC6A9S1PR3KCNH2BRD4
SCHEMBL5043148 0.80 MAPK1 (0.49) SLC6A9S1PR3SYK
SCHEMBL20476411 0.80 XDH (0.46) SLC6A9S1PR3
SCHEMBL5041677 0.78 FABP4 (0.45) SLC6A9S1PR3APEX1SYKFABP4
SCHEMBL17027246 0.77 PTGDR2 (0.50) PIM1PIM2APEX1SYKKMO
SCHEMBL5041907 0.77 PDE4A (0.42) SLC6A9MRGPRX1APEX1SYKFABP4
SCHEMBL4422191 0.77 APEX1 (0.44) SLC6A9S1PR3MRGPRX1APEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656361-B1 PIPERAZINE WITH OR-SUBSTITUTED PHENYL GROUP AND THEIR USE AS GLYT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed