SCHEMBL5046544

SCHEMBL5046544

C[CH]Cc1cccc(CO)c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.47
PRSS2 P07478 1/20 0.47
PRSS3 P35030 1/20 0.47
ENPP2 Q13822 1/20 0.45
TSHR P16473 1/20 0.42
PRKCI P41743 1/20 0.41
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
S1PR1 P21453 6/20 0.39
DAO P14920 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
NOS3 P29474 2/20 0.37
NOS1 P29475 2/20 0.37
NOS2 P35228 2/20 0.37
CFTR P13569 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9202795 0.89 MAOB (0.38) NOS3NOS1NOS2
SCHEMBL10661810 0.83 PRSS1 (0.48) PRSS1PRSS2PRSS3ENPP2TSHR
SCHEMBL10661820 0.83 PRSS1 (0.48) PRSS1PRSS2PRSS3ENPP2TSHR
SCHEMBL123838 0.81 TSHR (0.61) PRSS1PRSS2PRSS3ENPP2TSHR
SCHEMBL2811400 0.79 PRSS1 (0.44) PRSS1PRSS2PRSS3ENPP2TSHR
SCHEMBL3506161 0.78 ENPP2 (0.54) ENPP2
SCHEMBL27483739 0.78 PNMT (0.48) ENPP2MRGPRX4NOS3NOS1NOS2
SCHEMBL4872736 0.78 XDH (0.50) PRSS1PRSS2PRSS3ENPP2TSHR
Hydrochloric Acid SCHEMBL14334287 0.78 ENPP2 (0.58) PRSS1PRSS2PRSS3ENPP2TSHR
SCHEMBL5793223 0.76 TAAR1 (0.52) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716150-B1 SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE AMGEN INC (US) 2008-04-23 EP disclosed