SCHEMBL5046915

SCHEMBL5046915

CCOC(=O)n1ccc2cc(F)cc(NS(=O)(=O)c3cccs3)c21

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
TSHR P16473 1/20 0.48
CYP2C19 P33261 1/20 0.48
CNKSR1 Q969H4 4/20 0.46
AKT1 P31749 2/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPT P10636 2/20 0.46
TP53 P04637 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HIF1A Q16665 1/20 0.46
LMNA P02545 1/20 0.45
HPGD P15428 1/20 0.45
PLK1 P53350 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CCR2 P41597 1/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1653185 0.78 ALDH1A1 (0.44) ALDH1A1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL1653068 0.76 MEN1 (0.46) ALDH1A1CNKSR1AKT1MEN1KMT2A
SCHEMBL5046916 0.73 MAPT (0.47) ALDH1A1TSHRCNKSR1AKT1MEN1
SCHEMBL7570349 0.70 ALDH1A1 (0.60) ALDH1A1CNKSR1AKT1MEN1KMT2A
SCHEMBL2354908 0.70 MEN1 (0.53) ALDH1A1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL1654094 0.70 ALDH1A1 (0.50) ALDH1A1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL1652707 0.69 CNKSR1 (0.47) ALDH1A1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL12783356 0.69 MEN1 (0.49) ALDH1A1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL7571210 0.68 CCR2 (0.67) ALDH1A1MEN1KMT2AMAPTTP53
SCHEMBL1653233 0.68 MEN1 (0.45) ALDH1A1CYP3A4CYP2C9TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1873144-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2008-01-02 EP disclosed