SCHEMBL5047725

SCHEMBL5047725

CCOC(=O)C(OC)c1c(F)cc(-c2cc[n+]([O-])cc2)cc1F

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.33
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
TMPRSS2 O15393 1/20 0.32
F10 P00742 1/20 0.32
PRSS1 P07477 1/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
SRD5A2 P31213 1/20 0.31
PRKCZ Q05513 1/20 0.31
GAA P10253 1/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5045168 0.84 ALDH1A1 (0.36) LMNAALDH1A1MEN1KMT2AGAA
SCHEMBL5045404 0.82 CDC7 (0.41) ALDH1A1HPGD
SCHEMBL5040747 0.77 CA12 (0.42) GAAHPGD
SCHEMBL2341607 0.74 PTGS2 (0.39) ALDH1A1NPC1RAB9ATSHRMAPK1
Hydrochloric Acid SCHEMBL5040718 0.72 F2 (0.43) TMPRSS2F10PRSS1
SCHEMBL5041381 0.68 CA12 (0.36) ALDH1A1MEN1KMT2AGAAHPGD
SCHEMBL5045621 0.68 ROCK1 (0.37) PRSS1
SCHEMBL5042607 0.66 CYP3A4 (0.40) ALDH1A1MEN1KMT2APRKCZGAA
SCHEMBL5042392 0.65 CA12 (0.42) GAAHPGD
SCHEMBL5045318 0.65 FEN1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567498-B1 MANDELIC ACID DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-23 EP disclosed
US-7129238-B2 Mandelic acid derivatives HOFFMANN-LA ROCHE INC. (US) 2006-10-31 US disclosed
US-20040122057-A1 Novel mandelic acid derivatives HOFFMANN-LA ROCHE INC. 2004-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122057-A1 Novel mandelic acid derivatives F7, F11, F9 LMNA 1694/4885ALDH1A1 519/4885MEN1 766/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.