SCHEMBL5048004

SCHEMBL5048004

O=CC(OC(c1ccccc1)c1ccccc1)N1CCN(Cc2ccnc(Cl)c2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.41
KDM4E B2RXH2 1/20 0.40
TSHR P16473 1/20 0.40
CYP3A4 P08684 2/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
USP2 O75604 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
HPN P05981 1/20 0.40
CHRM2 P08172 1/20 0.40
ADRA2A P08913 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD2 P14416 1/20 0.40
ADRA2C P18825 1/20 0.40
CNR1 P21554 1/20 0.40
DRD1 P21728 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4279870 0.77 ALDH1A1 (0.52) ATMKDM4ETSHRCYP3A4MEN1
SCHEMBL5035553 0.72 DRD2 (0.51) DRD2DRD4DRD3LMNASMN1; SMN2
SCHEMBL7606866 0.70 SMN1; SMN2 (0.57) KDM4ECYP2D6CYP2C19SMN1; SMN2
SCHEMBL5251748 0.70 SIGMAR1 (0.53) ATMKDM4ETSHRDRD4MEN1
SCHEMBL23358024 0.69 RECQL (0.52) KDM4ESMN1; SMN2CCR2
SCHEMBL29944490 0.69 RECQL (0.52) KDM4ESMN1; SMN2CCR2
SCHEMBL937589 0.69 SMN1; SMN2 (0.54) KDM4ESMN1; SMN2
SCHEMBL31669110 0.69 SMN1; SMN2 (0.54) KDM4ESMN1; SMN2
SCHEMBL17331777 0.68 MC4R (0.54) KDM4ELMNA
SCHEMBL9262526 0.68 SIGMAR1 (0.50) ATMKDM4EDRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1976841-A1 HETEROCYCLIC AMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS Neuromed Pharmaceuticals, Ltd. (CA) 2008-10-08 EP claimed
WO-2007071035-A1 HETEROCYCLIC AMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2007-06-28 WO claimed