SCHEMBL5048124

SCHEMBL5048124

O=C(Nc1nc(Cl)c2ncn(C(Cc3ccccc3)C(=O)O)c2n1)OCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SCD O00767 2/20 0.39
ACHE P22303 2/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 1/20 0.38
POLB P06746 1/20 0.38
PTGER1 P34995 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MAPKAPK2 P49137 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
TSHR P16473 1/20 0.37
FSHR P23945 1/20 0.37
CTRB1 P17538 2/20 0.37
MGLL Q99685 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5051783 0.94 MAP3K5 (0.40) MAP3K5SMN1; SMN2SCDACHENPC1
SCHEMBL5050469 0.92 TRPV1 (0.41) MAP3K5SMN1; SMN2SCDACHENPC1
SCHEMBL5048107 0.87 ACHE (0.38) SMN1; SMN2ACHENPC1KDM4EMAPT
SCHEMBL7617736 0.87 SMN1; SMN2 (0.37) SMN1; SMN2ACHENPC1POLBKDM4E
SCHEMBL5045348 0.85 ACHE (0.37) ACHENPC1KDM4EMAPTTDP1
SCHEMBL7843904 0.80 SCD (0.43) SMN1; SMN2SCDACHENPC1RAB9A
SCHEMBL9079905 0.79 MEN1 (0.42) MAP3K5SMN1; SMN2SCDACHEPTGER1
SCHEMBL7617492 0.79 HDAC1 (0.45) POLBKDM4EMAPTTDP1
SCHEMBL14309812 0.74 TSHR (0.43) SMN1; SMN2ACHENPC1RAB9APOLB
SCHEMBL14477481 0.73 RAB9A (0.46) SMN1; SMN2ACHENPC1RAB9APTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1873156-A1 Process for the preparation of 6-[[(alkoxy)carbonyl]amino]-9H-Purine-9-acetic acid and 4-[(alkoxycarbonyl)amino]-2-oxo-1(2H)-Pyrimidineacetic acid derivatives as synthons for the synthesis of peptide nucleic acids PerSeptive Biosystems, Inc. (US) 2008-01-02 EP disclosed
EP-0736027-B1 GUANINE SYNTHONS FOR PEPTIDE NUCLEIC ACID SYNTHESIS AND METHOD FOR PRODUCTION PERSEPTIVE BIOSYSTEMS INC (US) 2002-05-29 EP disclosed